195
|
639
|
7k7zA |
Structure of a hit for g protein coupled receptor kinase 2 (grk2) inhibitor for the potential treatment of heart failure |
75
|
266
|
7ayhA |
Crystal structure of aurora a in complex with 7-(2-anilinopyrimidin-4-yl)-1-benzazepin-2-one derivative (compound 2c) |
98
|
322
|
6z3uB |
Structure of the cak complex form chaetomium thermophilum |
81
|
281
|
7b31A |
Mst3 in complex with compound mria9 |
117
|
328
|
7a1zA |
Crystal structure of human protein kinase ck2alpha' (csnk2a2 gene product) in complex with the atp-competitive inhibitor 6-bromo-5-chloro-1h-triazolo[4,5-b]pyridine |
102
|
322
|
6z4xB |
Structure of the cak complex form chaetomium thermophilum bound to atp-gamma-s |
79
|
279
|
7b35A |
Mst3 in complex with compound mria13 |
90
|
293
|
7akgA |
Crystal structure of stk17b with bound dovitinib |
111
|
350
|
6zqsA |
Crystal structure of double-phosphorylated p38alpha with atf2(83-102) |
85
|
283
|
7b36A |
Mst4 in complex with compound g-5555 |
90
|
360
|
6zr5A |
Crystal structure of jnk1 in complex with atf2(19-58) |
72
|
298
|
7kacA |
Crystal structure of hpk1 (map4k1) kinase in complex with 5-{[4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-5-(1,3,4-oxadiazol-2-yl)pyrimidin-2-yl]amino}-3,3-dimethyl-2-benzofuran-1(3h)-one |
99
|
347
|
7b6fA |
Gsk3-beta in complex with compound (s)-5c |
115
|
334
|
7a49A |
Crystal structure of human protein kinase ck2alpha (csnk2a1 gene product) in complex with the atp-competitive inhibitor 6-bromo-5-chloro-1h-triazolo[4,5-b]pyridine |
78
|
268
|
7ayiA |
Crystal structure of aurora a in complex with 7-(2-anilinopyrimidin-4-yl)-1-benzazepin-2-one derivative (compound 2a) |
85
|
281
|
7b32A |
Mst3 in complex with mria7 |
89
|
268
|
6xoeA |
Cocrystal structure of human camkii-alpha (camk2a)kinase domain and glun2b(s1303d) in complex with atp |
81
|
268
|
7kl1A |
Cocrystal structure of human camkii-alpha (camk2a)kinase domain and glun2b(s1303d) in complex with atp |
113
|
327
|
7a1bA |
Crystal structure of human protein kinase ck2alpha' (csnk2a2 gene product) in complex with the atp-competitive inhibitor 5,6-dibromo-1h-triazolo[4,5-b]pyridine |
109
|
338
|
6z08A |
Crystal structure of camp-dependent protein kinase a (cho pka) in complex with 4-nitrophenol |
115
|
325
|
7a2hA |
Crystal structure of human protein kinase ck2alpha' (csnk2a2 gene product) in complex with the atp-competitive inhibitor 5,6,7-tribromo-1h-imidazo[4,5-b]pyridine |
110
|
338
|
6zn0A |
Crystal structure of camp-dependent protein kinase a (cho pka) in complex with isonicotinamidine |
112
|
333
|
7a4bA |
Crystal structure of human protein kinase ck2alpha (csnk2a1 gene product) in complex with the atp-competitive inhibitor 5,6-dibromo-1h-triazolo[4,5-b]pyridine |
122
|
333
|
6tluAAA |
Human ck2 kinase alpha subunit in complex with the atp-competitive inhibitor 4,5-dibromobenzotriazole |
129
|
333
|
6tlsA |
Human ck2 kinase alpha subunit in complex with the atp-competitive inhibitor 4,6-dibromobenzotriazole |
83
|
273
|
6vruA |
Pim-inhibitor complex 1 |
94
|
401
|
6w3eA |
Structure of phosphorylated ire1 in complex with g-0701 |
127
|
402
|
6w3kA |
Structure of unphosphorylated human ire1 bound to g-9807 |
83
|
268
|
6x8vA |
Cocrystal structure of human camkii-alpha (camk2a)kinase domain and tiam1 |
79
|
268
|
6xbxA |
Cocrystal structure of human camkii-alpha (camk2a)kinase domain and glun2b in complex with atp |
86
|
267
|
6x5qA |
Cocrystal structure of human camkii-alpha (camk2a)kinase domain and glua1 |
128
|
402
|
6w3bA |
Structure of apo unphosphorylated ire1 |
90
|
344
|
6v2wB |
Crystal structure of the braf:mek1 kinases in complex with amppnp |
90
|
342
|
6v31B |
Crystal structure of the braf:mek1 kinases in complex with amppnp and ch5126766 |
82
|
271
|
6vrvA |
Discovery of sarxxxx92, a pan-pim kinase inhibitor, efficacious in a kg1 tumor model |
96
|
403
|
6w3aA |
Structure of unphosphorylated ire1 in complex with g-7658 |
88
|
324
|
6z45A |
Cdk9-cyclin-t1 complex bound by compound 24 |
94
|
342
|
6v2zB |
Crystal structure of the braf:mek1 kinases in complex with amppnp and cobimetinib |
125
|
405
|
6w3cA |
Structure of phosphorylated apo ire1 |
122
|
401
|
6w39A |
Structure of unphosphorylated ire1 in complex with g-1749 |
92
|
268
|
6x5gA |
Cocrystal structure of human camkii-alpha (camk2a)kinase domain and lrrc7 inhibitory domain |
98
|
346
|
6v2vB |
Crystal structure of the braf:mek1 kinases in complex with amppnp and pd0325901 |
86
|
343
|
6v2xB |
Crystal structure of the braf:mek1 kinases in complex with amppnp and binimetinib |
128
|
333
|
6tlvA |
Human ck2 kinase alpha subunit in complex with the atp-competitive inhibitor 5-bromobenzotriazole |
71
|
405
|
6wjfA |
Pka riibeta holoenzyme with dnajb1-pkac fusion in fibrolamellar hepatoceullar carcinoma |
126
|
333
|
6tloA |
Human ck2 kinase alpha subunit in complex with the atp-competitive inhibitor 4,5,6-tribromobenzotriazole |
88
|
344
|
6v30B |
Crystal structure of the braf:mek1 kinases in complex with amppnp and pimasertib |
93
|
268
|
6xdlA |
Cocrystal structure of human camkii-alpha (camk2a)kinase domain and glun2b |
88
|
340
|
6v2yB |
Crystal structure of the braf:mek1 kinases in complex with amppnp and trametinib |
48
|
310
|
6wjgA |
Pka riibeta holoenzyme with dnajb1-pkac fusion in fibrolamellar hepatoceullar carcinoma |