Found 159 chains in Genus chains table. Displaying 1 - 50. Applied filters: Proteins

Search results query: transcription/transcription inhibitor

Total Genus Sequence Length pdb Title
48 225 6cdyA Crystal structure of tead complexed with its inhibitor
47 225 6uybA Crystal structure of tead2 bound to compound 1
185 552 6nuqA Stat3 core in complex with compound si109
183 552 6njsA Stat3 core in complex with compound sd36
98 268 6o67A Crystal structure of human ppargamma ligand binding domain in complex with mitoglitazone
91 270 6o68A Crystal structure of human ppargamma ligand binding domain in complex with ciglitazone
38 127 6mh1A Crystal structure of the first bromodomain of human brd4 in complex with hu-10, a 1,4,5-trisubstituted imidazole analogue
0 4 5x54C Crystal structure of the keap1 kelch domain in complex with a tetrapeptide
0 4 3pslC Fine-tuning the stimulation of mll1 methyltransferase activity by a histone h3 based peptide mimetic
42 109 6moaA C-terminal bromodomain of human brd2 in complex with 4-(2-cyclopropyl-7-(6-methylquinolin-5-yl)-1h-benzo[d]imidazol-5-yl)-3,5-dimethylisoxazole inhibitor
41 114 6mo7A N-terminal bromodomain of human brd2 with n-((4-(3-(n-cyclopentylsulfamoyl)-4-methylphenyl)-3-methylisoxazol-5-yl)methyl)acetamide inhibitor
41 114 6mo9A N-terminal bromodomain of human brd2 in complex with n-cyclopentyl-7-(3,5-dimethylisoxazol-4-yl)quinoline-5-sulfonamide inhibitor
42 114 6mo8A N-terminal bromodomain of human brd2 in complex with 4,4'-(quinoline-5,7-diyl)bis(3,5-dimethylisoxazole) inhibitor
97 268 6md2A Crystal structure of human ppargamma ligand binding domain in complex with gw9662 and arachidonic acid
98 268 6md4A Crystal structure of human ppargamma ligand binding domain in complex with rosiglitazone and oleic acid
76 333 6e3sB Crystal structure of the heterodimeric hif-2 complex with antagonist pt2385
68 328 6e3tB Crystal structure of the heterodimeric hif-2 complex with antagonist t1001
57 361 6e3tA Crystal structure of the heterodimeric hif-2 complex with antagonist t1001
41 127 6dmjA A multiconformer ligand model of inhibitor 53w bound to creb binding protein bromodomain
42 127 6dmlA A multiconformer ligand model of 3,5 dimethylisoxaxole bound to the bromodomain of human brd4
40 113 6dmkA A multiconformer ligand model of an isoxazolyl-benzimidazole ligand bound to the bromodomain of human crebbp
93 270 6dhaA Crystal structure of human ppargamma ligand binding domain in complex with hydroxy pioglitazone (m-iv)
72 367 6e3sA Crystal structure of the heterodimeric hif-2 complex with antagonist pt2385
83 242 6owcA Mutant estrogen receptor alpha (era) y537s covalently bound to h3b-6545.
100 270 6dgqA Crystal structure of human ppargamma ligand binding domain in complex with cay10506
95 270 6dh9A Crystal structure of human ppargamma ligand binding domain in complex with msdc-0602
103 270 6dgrA Crystal structure of human ppargamma ligand binding domain in complex with cay10638
97 270 6dglA Crystal structure of human ppargamma ligand binding domain in complex with darglitazone
94 268 6dgoA Crystal structure of human ppargamma ligand binding domain in complex with troglitazone
38 110 5jwmA Bivalent bet bromodomain inhibition
58 210 5ke3A Crystal structure of setdb1 tudor domain in complex with fragment mrt0181a
51 180 5h1uA Complex structure of trim24 phd-bromodomain and inhibitor 2
48 127 5hclA Crystal structure of the first bromodomain of brd4 in complex with dma
50 182 5h1tA Complex structure of trim24 phd-bromodomain and inhibitor 1
320 1340 4yfnC Escherichia coli rna polymerase in complex with squaramide compound 14 (n-[3,4-dioxo-2-(4-{[4-(trifluoromethyl)benzyl]amino}piperidin-1-yl)cyclobut-1-en-1-yl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide)
309 1369 4yfkD Escherichia coli rna polymerase in complex with squaramide compound 8.
40 229 4yfxA Escherichia coli rna polymerase in complex with myxopyronin b
23 89 4yfnE Escherichia coli rna polymerase in complex with squaramide compound 14 (n-[3,4-dioxo-2-(4-{[4-(trifluoromethyl)benzyl]amino}piperidin-1-yl)cyclobut-1-en-1-yl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide)
39 112 6c7qA Brd4 bd2 in complex with compound ce277
34 108 6c7rA Brd4 bd1 in complex with compound cf53
82 228 6bn6A Identification of bicyclic hexafluoroisopropyl alcohol sulfonamides as rorgt/rorc inverse agonists
85 240 5wgqA Estrogen receptor alpha ligand binding domain in complex with estradiol and src2-bcp1
36 127 5wmgA N-terminal bromodomain of brd4 in complex with otx-015
42 109 5u6vA X-ray crystal structure of 1,2,3-triazolobenzodiazepine in complex with brd2(d2)
40 127 5wmdA N-terminal bromodomain of brd4 in complex with otx-015
93 241 5c4tA Identification of a novel allosteric binding site for rorgt inhibitors
92 241 5c4oA Identification of a novel allosteric binding site for rorgt inhibitors
317 1340 4yfkC Escherichia coli rna polymerase in complex with squaramide compound 8.
52 183 4ybmA Crystal structure of trim24 phd-bromodomain complexed with n-{6-[3-(benzyloxy)phenoxy]-1,3-dimethyl-2-oxo-2,3-dihydro-1h-1,3-benzodiazol-5-yl}-3,4-dimethoxybenzene-1-sulfonamide (7b)
57 319 4yfkA Escherichia coli rna polymerase in complex with squaramide compound 8.