2WAPA

3d-crystal structure of humanized-rat fatty acid amide hydrolase (faah) conjugated with the drug-like urea inhibitor pf-3845
Total Genus 221
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The genus trace: a function that shows values of genus (vertical axis) for subchains spanned between the first residue, and all other residues (shown on horizontal axis). The number of the latter residue and the genus of a given subchain are shown interactively.

Total Genus
221
sequence length
541
structure length
541
Chain Sequence
GRQKARGAATRARQKQRASLETMDKAVQRFRLQNPDLDSEALLTLPLLQLVQKLQSGELSPEAVFFTYLGKAWEVNKGTNCVTSYLTDCETQLSQAPRQGLLYGVPVSLKECFSYKGHDSTLGLSLNEGMPSESDCVVVQVLKLQGAVPFVHTNVPQSMFSYDCSNPLFGQTMNPWKSSKSPGGSSGGEGALIGSGGSPLGLGTDIGGSIRFPSAFCGICGLKPTGNRLSKSGLKGCVYGQTAVQLSLGPMARDVESLALCLKALLCEHLFTLDPTVPPLPFREEVYRSSRPLRVGYYETDNYTMPSPAMRRALIETKQRLEAAGHTLIPFLPNNIPYALEVLSTGGLFSDGGRSFLQNFKGDFVDPCLGDLILILRLPSWFKRLLSLLLKPLFPRLAAFLNNMRPRSAEKLWKLQHEIEMYRQSVIAQWKAMNLDVLLTPMLGPALDLNTPGRATGAVSYTMLYNCLDFPAGVVPVTTVTAEDDAQMELYKGYFGDIWDIILKKAMKNSVGLPVAVQCVALPWQEELCLRFMREVEQLMT
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The genus matrix. At position (x,y) a genus value for a subchain spanned between x’th and y’th residue is shown. Values of the genus are represented by color, according to the scale given on the right.

Structure visualization

After clicking on a point (x,y) in the genus matrix above, a subchain from x to y is shown in color.

molecule tags Hydrolase
molecule keywords FATTY-ACID AMIDE HYDROLASE 1
publication title Discovery and Characterization of a Highly Selective Faah Inhibitor that Reduces Inflammatory Pain.
pubmed doi rcsb
source organism Rattus norvegicus
total genus 221
structure length 541
sequence length 541
chains with identical sequence B
ec nomenclature ec 3.5.1.99: Fatty acid amide hydrolase.
pdb deposition date 2009-02-11

pfam database annotations

chain Pfam Accession Code Pfam Family Identifier Pfam Description
A PF01425 Amidase Amidase
Image from the rcsb pdb (www.rcsb.org)
cath code
ClassArchitectureTopologyHomologyDomain
3.90.1300.10 Alpha Beta Alpha-Beta Complex Amidase signature (AS) enzymes Amidase signature (AS) domain 2wapA00
2G5IA 3OJ8A 3QKVA 1O9QA 4ISTA 1M22A 1OBKA 4GYSA 2VYAA 2WJ1A 3PR0A 1OBLA 3QJ9A 4GYRA 3KFUE 4J5PA 3K83A 4YJIA 2WAPA 5EWQA 1OCHA 3A1KA 1OCKA 1OBJA 3K7FA 3K84A 2F2AA 3H0LA 1OCMA 3H0MA 3QJ8A 4WJ3A 1O9NA 3IP4A 2WJ2A 4YJ6A 1OCLA 1O9OA 2GI3A 2DQNA 3AL0A 3A2PA 1MT5A 4N0IA 1OBIA 2G5HA 3A2QA 3LJ7A 1O9PA 4ISSA 2DF4A 5AC3A 2DC0A 3LJ6A 3H0RA 4N0HA 4HBPA 1M21A 3A1IA 3PPMA 3QK5A 4CP8A 4DO3A
chains in the Genus database with same CATH superfamily
2G5IA 3OJ8A 3QKVA 1O9QA 4ISTA 1M22A 1OBKA 4GYSA 2VYAA 2WJ1A 3PR0A 1OBLA 3QJ9A 4GYRA 3KFUE 4J5PA 3K83A 4YJIA 2WAPA 5EWQA 1OCHA 3A1KA 1OCKA 1OBJA 3K7FA 3K84A 2F2AA 3H0LA 1OCMA 3H0MA 3QJ8A 4WJ3A 1O9NA 3IP4A 2WJ2A 4YJ6A 1OCLA 1O9OA 2GI3A 2DQNA 3AL0A 3A2PA 1MT5A 4N0IA 1OBIA 2G5HA 3A2QA 3LJ7A 1O9PA 4ISSA 2DF4A 5AC3A 2DC0A 3LJ6A 3H0RA 4N0HA 4HBPA 1M21A 3A1IA 3PPMA 3QK5A 4CP8A 4DO3A
chains in the Genus database with same CATH topology
2G5IA 3OJ8A 3QKVA 1O9QA 4ISTA 1M22A 1OBKA 4GYSA 2VYAA 2WJ1A 3PR0A 1OBLA 3QJ9A 4GYRA 3KFUE 4J5PA 3K83A 4YJIA 2WAPA 5EWQA 1OCHA 3A1KA 1OCKA 1OBJA 3K7FA 3K84A 2F2AA 3H0LA 1OCMA 3H0MA 3QJ8A 4WJ3A 1O9NA 3IP4A 2WJ2A 4YJ6A 1OCLA 1O9OA 2GI3A 2DQNA 3AL0A 3A2PA 1MT5A 4N0IA 1OBIA 2G5HA 3A2QA 3LJ7A 1O9PA 4ISSA 2DF4A 5AC3A 2DC0A 3LJ6A 3H0RA 4N0HA 4HBPA 1M21A 3A1IA 3PPMA 3QK5A 4CP8A 4DO3A
chains in the Genus database with same CATH homology


 
#chains in the Genus database with same CATH superfamily
 2G5I A;  3OJ8 A;  3QKV A;  1O9Q A;  4IST A;  1M22 A;  1OBK A;  4GYS A;  2VYA A;  2WJ1 A;  3PR0 A;  1OBL A;  3QJ9 A;  4GYR A;  3KFU E;  4J5P A;  3K83 A;  4YJI A;  2WAP A;  5EWQ A;  1OCH A;  3A1K A;  1OCK A;  1OBJ A;  3K7F A;  3K84 A;  2F2A A;  3H0L A;  1OCM A;  3H0M A;  3QJ8 A;  4WJ3 A;  1O9N A;  3IP4 A;  2WJ2 A;  4YJ6 A;  1OCL A;  1O9O A;  2GI3 A;  2DQN A;  3AL0 A;  3A2P A;  1MT5 A;  4N0I A;  1OBI A;  2G5H A;  3A2Q A;  3LJ7 A;  1O9P A;  4ISS A;  2DF4 A;  5AC3 A;  2DC0 A;  3LJ6 A;  3H0R A;  4N0H A;  4HBP A;  1M21 A;  3A1I A;  3PPM A;  3QK5 A;  4CP8 A;  4DO3 A; 
#chains in the Genus database with same CATH topology
 2G5I A;  3OJ8 A;  3QKV A;  1O9Q A;  4IST A;  1M22 A;  1OBK A;  4GYS A;  2VYA A;  2WJ1 A;  3PR0 A;  1OBL A;  3QJ9 A;  4GYR A;  3KFU E;  4J5P A;  3K83 A;  4YJI A;  2WAP A;  5EWQ A;  1OCH A;  3A1K A;  1OCK A;  1OBJ A;  3K7F A;  3K84 A;  2F2A A;  3H0L A;  1OCM A;  3H0M A;  3QJ8 A;  4WJ3 A;  1O9N A;  3IP4 A;  2WJ2 A;  4YJ6 A;  1OCL A;  1O9O A;  2GI3 A;  2DQN A;  3AL0 A;  3A2P A;  1MT5 A;  4N0I A;  1OBI A;  2G5H A;  3A2Q A;  3LJ7 A;  1O9P A;  4ISS A;  2DF4 A;  5AC3 A;  2DC0 A;  3LJ6 A;  3H0R A;  4N0H A;  4HBP A;  1M21 A;  3A1I A;  3PPM A;  3QK5 A;  4CP8 A;  4DO3 A; 
#chains in the Genus database with same CATH homology
 2G5I A;  3OJ8 A;  3QKV A;  1O9Q A;  4IST A;  1M22 A;  1OBK A;  4GYS A;  2VYA A;  2WJ1 A;  3PR0 A;  1OBL A;  3QJ9 A;  4GYR A;  3KFU E;  4J5P A;  3K83 A;  4YJI A;  2WAP A;  5EWQ A;  1OCH A;  3A1K A;  1OCK A;  1OBJ A;  3K7F A;  3K84 A;  2F2A A;  3H0L A;  1OCM A;  3H0M A;  3QJ8 A;  4WJ3 A;  1O9N A;  3IP4 A;  2WJ2 A;  4YJ6 A;  1OCL A;  1O9O A;  2GI3 A;  2DQN A;  3AL0 A;  3A2P A;  1MT5 A;  4N0I A;  1OBI A;  2G5H A;  3A2Q A;  3LJ7 A;  1O9P A;  4ISS A;  2DF4 A;  5AC3 A;  2DC0 A;  3LJ6 A;  3H0R A;  4N0H A;  4HBP A;  1M21 A;  3A1I A;  3PPM A;  3QK5 A;  4CP8 A;  4DO3 A; 
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similar chains in the Genus database (?% sequence similarity)
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similar chains in the pdb database (?% sequence similarity)

 
#similar chains in the Genus database (?% sequence similarity)
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#similar chains, but unknotted
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