4L2GC

Tankyrase 2 in complex with 6- fluoro flavone
Total Genus 1
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The genus trace: a function that shows values of genus (vertical axis) for subchains spanned between the first residue, and all other residues (shown on horizontal axis). The number of the latter residue and the genus of a given subchain are shown interactively.

Total Genus
1
sequence length
47
structure length
47
Chain Sequence
MAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE
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The genus matrix. At position (x,y) a genus value for a subchain spanned between x’th and y’th residue is shown. Values of the genus are represented by color, according to the scale given on the right.

Structure visualization

After clicking on a point (x,y) in the genus matrix above, a subchain from x to y is shown in color.

molecule tags Transferase/transferase inhibitor
molecule keywords Tankyrase-2
publication title Discovery of tankyrase inhibiting flavones with increased potency and isoenzyme selectivity.
pubmed doi rcsb
source organism Homo sapiens
total genus 1
structure length 47
sequence length 47
chains with identical sequence D
ec nomenclature ec 2.4.2.30: NAD(+) ADP-ribosyltransferase.
pdb deposition date 2013-06-04
Image from the rcsb pdb (www.rcsb.org)
cath code
ClassArchitectureTopologyHomologyDomain
3.40.1620.50 Alpha Beta 3-Layer(aba) Sandwich YefM-like fold YefM-like fold 4l2gC00
4UVPB 4UI6C 4HKNC 4UI8C 4L32C 4L2GC 4L0IC 4UI4C 4HLFC 4L31C 4L33C 4L2FC 4UI5C 4L10C 5ADTB 4HMHC 4L0BC 4HKIC 4L34C 5C5RC 5ADQB 4UI3C 4KZQC 4KZUC 5C5QC 4UI7C 5FPFC 4L09C 4L0VC 4HLKC 4HLGC 4HKKB 4KZLC 4L0TC 4L0SC 5ADSB 5C5PC 4HL5C 5ADRB 4HLMC 4HLHC 4L2KC
chains in the Genus database with same CATH superfamily
4UVPB 4ZLXA 4UI6C 4HKNC 4UI8C 3K6QA 4L32C 4L0IC 4L2GC 4UI4C 4HLFC 4L31C 3OEIE 2A6QA 3G5OA 4L33C 4L2FC 4UI5C 4L10C 4ZM2A 5ADTB 3OEIA 4HMHC 4L0BC 4ZM0A 4HKIC 4L34C 5C5RC 5ADQB 4UI3C 3HRYA 2ZIXB 4KZQC 4KZUC 5C5QC 3D55A 4UI7C 5FPFC 4L09C 3HJ6A 4L0VC 4HLKC 3CTOA 2ODKA 4HLGC 4HKKB 4KZLC 4L0TC 3K33B 3KH2E 4L0SC 5ADSB 5C5PC 4HL5C 5ADRB 4HLMC 3HS2A 4HLHC 4L2KC
chains in the Genus database with same CATH topology
4UVPB 4UI6C 4HKNC 4UI8C 4L32C 4L2GC 4L0IC 4UI4C 4HLFC 4L31C 4L33C 4L2FC 4UI5C 4L10C 5ADTB 4HMHC 4L0BC 4HKIC 4L34C 5C5RC 5ADQB 4UI3C 2ZIXB 4KZQC 4KZUC 5C5QC 4UI7C 5FPFC 4L09C 3HJ6A 4L0VC 4HLKC 4HLGC 4HKKB 4KZLC 4L0TC 4L0SC 5ADSB 5C5PC 4HL5C 5ADRB 4HLMC 4HLHC 4L2KC
chains in the Genus database with same CATH homology


 
#chains in the Genus database with same CATH superfamily
 4UVP B;  4UI6 C;  4HKN C;  4UI8 C;  4L32 C;  4L2G C;  4L0I C;  4UI4 C;  4HLF C;  4L31 C;  4L33 C;  4L2F C;  4UI5 C;  4L10 C;  5ADT B;  4HMH C;  4L0B C;  4HKI C;  4L34 C;  5C5R C;  5ADQ B;  4UI3 C;  4KZQ C;  4KZU C;  5C5Q C;  4UI7 C;  5FPF C;  4L09 C;  4L0V C;  4HLK C;  4HLG C;  4HKK B;  4KZL C;  4L0T C;  4L0S C;  5ADS B;  5C5P C;  4HL5 C;  5ADR B;  4HLM C;  4HLH C;  4L2K C; 
#chains in the Genus database with same CATH topology
 4UVP B;  4ZLX A;  4UI6 C;  4HKN C;  4UI8 C;  3K6Q A;  4L32 C;  4L0I C;  4L2G C;  4UI4 C;  4HLF C;  4L31 C;  3OEI E;  2A6Q A;  3G5O A;  4L33 C;  4L2F C;  4UI5 C;  4L10 C;  4ZM2 A;  5ADT B;  3OEI A;  4HMH C;  4L0B C;  4ZM0 A;  4HKI C;  4L34 C;  5C5R C;  5ADQ B;  4UI3 C;  3HRY A;  2ZIX B;  4KZQ C;  4KZU C;  5C5Q C;  3D55 A;  4UI7 C;  5FPF C;  4L09 C;  3HJ6 A;  4L0V C;  4HLK C;  3CTO A;  2ODK A;  4HLG C;  4HKK B;  4KZL C;  4L0T C;  3K33 B;  3KH2 E;  4L0S C;  5ADS B;  5C5P C;  4HL5 C;  5ADR B;  4HLM C;  3HS2 A;  4HLH C;  4L2K C; 
#chains in the Genus database with same CATH homology
 4UVP B;  4UI6 C;  4HKN C;  4UI8 C;  4L32 C;  4L2G C;  4L0I C;  4UI4 C;  4HLF C;  4L31 C;  4L33 C;  4L2F C;  4UI5 C;  4L10 C;  5ADT B;  4HMH C;  4L0B C;  4HKI C;  4L34 C;  5C5R C;  5ADQ B;  4UI3 C;  2ZIX B;  4KZQ C;  4KZU C;  5C5Q C;  4UI7 C;  5FPF C;  4L09 C;  3HJ6 A;  4L0V C;  4HLK C;  4HLG C;  4HKK B;  4KZL C;  4L0T C;  4L0S C;  5ADS B;  5C5P C;  4HL5 C;  5ADR B;  4HLM C;  4HLH C;  4L2K C; 
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similar chains in the Genus database (?% sequence similarity)
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similar chains in the pdb database (?% sequence similarity)

 
#similar chains in the Genus database (?% sequence similarity)
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#similar chains, but unknotted
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#similar chains in the pdb database (?% sequence similarity)
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