4ZTVA

Non-anthranilate-like inhibitor (tamu-a7) complexed with anthranilate phosphoribosyltransferase (trpd) from mycobacterium tuberculosis in absence of prpp
Total Genus 124
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The genus trace: a function that shows values of genus (vertical axis) for subchains spanned between the first residue, and all other residues (shown on horizontal axis). The number of the latter residue and the genus of a given subchain are shown interactively.

Total Genus
124
sequence length
347
structure length
339
Chain Sequence
PSWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGNTVNLSTMAAIVVAAAGVPVVKHGNRASGGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSRAEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQIL
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The genus matrix. At position (x,y) a genus value for a subchain spanned between x’th and y’th residue is shown. Values of the genus are represented by color, according to the scale given on the right.

Structure visualization

After clicking on a point (x,y) in the genus matrix above, a subchain from x to y is shown in color.

Chord Diagram
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molecule tags Transferase/transferase inhibitor
molecule keywords Anthranilate phosphoribosyltransferase
publication title Bioactive non-anthranilate-like fragment-like inhibitor provides alternative starting point for inhibitor design against anthranilate phosphoribosyl transferase from Mycobacterium tuberculosis.
rcsb
source organism Mycobacterium tuberculosis
total genus 124
structure length 339
sequence length 347
chains with identical sequence B
ec nomenclature ec 2.4.2.18: Anthranilate phosphoribosyltransferase.
pdb deposition date 2015-05-15

pfam database annotations

chain Pfam Accession Code Pfam Family Identifier Pfam Description
A PF00591 Glycos_transf_3 Glycosyl transferase family, a/b domain
A PF02885 Glycos_trans_3N Glycosyl transferase family, helical bundle domain
Image from the rcsb pdb (www.rcsb.org)
cath code
ClassArchitectureTopologyHomologyDomain
1.20.970.10 Mainly Alpha Up-down Bundle Transferase, Pyrimidine Nucleoside Phosphorylase; Chain A, domain 3 Transferase, Pyrimidine Nucleoside Phosphorylase; Chain C 4ztvA01
3.40.1030.10 Alpha Beta 3-Layer(aba) Sandwich Pyrimidine Nucleoside Phosphorylase; Chain A, domain 2 Nucleoside phosphorylase/phosphoribosyltransferase catalytic domain 4ztvA02
5BNEA 4X58A 1O17A 4YI7A 4X46A 4LHMA 4GA4A 4YEKA 4X5DA 3QR9A 1ZVWA 5EP8A 3H5QA 3GBRA 3QSAA 4X5AA 2TPTA 4N5VA 5BO2A 4X59A 4ZOJA 5EY3A 5C7SA 2ELCA 4EAFA 4GIUA 2WK5A 4OWMA 1ZYKA 4ZOFA 4EADA 1BRWA 4N8QA 1AZYA 3TWPA 4OWUA 4ZOKA 4M0RA 4OWVA 2GVQA 4N93A 5C2LA 2BPQA 1GXBA 4X5BA 1ZXYA 4GA5A 4HKMA 5C1RA 4YYYA 4OWOA 5BO3A 3UU1A 2DSJA 4ZTVA 5BYTA 4MUOA 4GA6A 2WK6A 4IJ1A 4XR5A 3QS8A 2J0FA 1V8GA 1VQUA 4OWNA 4GTNA 1KGZA 3QQSA 3R88A 4OWQA 4GKMA 4X5CA 4OWSA 1KHDA 1UOUA 4X5EA 1OTPA 3R6CA
chains in the Genus database with same CATH superfamily
5BNEA 4X58A 1O17A 4YI7A 4X46A 4LHMA 4GA4A 4YEKA 4X5DA 3QR9A 1ZVWA 5EP8A 3H5QA 3GBRA 3QSAA 4X5AA 2TPTA 4N5VA 5BO2A 4X59A 4ZOJA 5EY3A 1RRZA 5C7SA 2ELCA 4EAFA 4GIUA 2WK5A 4OWMA 1ZYKA 4ZOFA 4EADA 1BRWA 4N8QA 1AZYA 3TWPA 4OWUA 4ZOKA 4F3FC 4M0RA 4OWVA 2GVQA 4N93A 5C2LA 2BPQA 1GXBA 4X5BA 1ZXYA 4GA5A 4HKMA 5C1RA 4YYYA 4OWOA 5BO3A 3UU1A 2DSJA 4ZTVA 5BYTA 4MUOA 4GA6A 2WK6A 4IJ1A 4XR5A 3QS8A 2J0FA 1V8GA 1VQUA 4OWNA 4GTNA 1KGZA 3QQSA 3R88A 4OWQA 4GKMA 4X5CA 1RF8B 4OWSA 1KHDA 1UOUA 4X5EA 1OTPA 3R6CA
chains in the Genus database with same CATH topology
5BNEA 4X58A 1O17A 4YI7A 4X46A 4LHMA 4GA4A 4YEKA 4X5DA 3QR9A 1ZVWA 5EP8A 3H5QA 3GBRA 3QSAA 4X5AA 2TPTA 4N5VA 5BO2A 4X59A 4ZOJA 5EY3A 5C7SA 2ELCA 4EAFA 4GIUA 2WK5A 4OWMA 1ZYKA 4ZOFA 4EADA 1BRWA 4N8QA 1AZYA 3TWPA 4OWUA 4ZOKA 4M0RA 4OWVA 2GVQA 4N93A 5C2LA 2BPQA 1GXBA 4X5BA 1ZXYA 4GA5A 4HKMA 5C1RA 4YYYA 4OWOA 5BO3A 3UU1A 2DSJA 4ZTVA 5BYTA 4MUOA 4GA6A 2WK6A 4IJ1A 4XR5A 3QS8A 2J0FA 1V8GA 1VQUA 4OWNA 4GTNA 1KGZA 3QQSA 3R88A 4OWQA 4GKMA 4X5CA 4OWSA 1KHDA 1UOUA 4X5EA 1OTPA 3R6CA
chains in the Genus database with same CATH homology


 
#chains in the Genus database with same CATH superfamily
 5BNE A;  4X58 A;  1O17 A;  4YI7 A;  4X46 A;  4LHM A;  4GA4 A;  4YEK A;  4X5D A;  3QR9 A;  1ZVW A;  5EP8 A;  3H5Q A;  3GBR A;  3QSA A;  4X5A A;  2TPT A;  4N5V A;  5BO2 A;  4X59 A;  4ZOJ A;  5EY3 A;  5C7S A;  2ELC A;  4EAF A;  4GIU A;  2WK5 A;  4OWM A;  1ZYK A;  4ZOF A;  4EAD A;  1BRW A;  4N8Q A;  1AZY A;  3TWP A;  4OWU A;  4ZOK A;  4M0R A;  4OWV A;  2GVQ A;  4N93 A;  5C2L A;  2BPQ A;  1GXB A;  4X5B A;  1ZXY A;  4GA5 A;  4HKM A;  5C1R A;  4YYY A;  4OWO A;  5BO3 A;  3UU1 A;  2DSJ A;  4ZTV A;  5BYT A;  4MUO A;  4GA6 A;  2WK6 A;  4IJ1 A;  4XR5 A;  3QS8 A;  2J0F A;  1V8G A;  1VQU A;  4OWN A;  4GTN A;  1KGZ A;  3QQS A;  3R88 A;  4OWQ A;  4GKM A;  4X5C A;  4OWS A;  1KHD A;  1UOU A;  4X5E A;  1OTP A;  3R6C A; 
#chains in the Genus database with same CATH topology
 5BNE A;  4X58 A;  1O17 A;  4YI7 A;  4X46 A;  4LHM A;  4GA4 A;  4YEK A;  4X5D A;  3QR9 A;  1ZVW A;  5EP8 A;  3H5Q A;  3GBR A;  3QSA A;  4X5A A;  2TPT A;  4N5V A;  5BO2 A;  4X59 A;  4ZOJ A;  5EY3 A;  1RRZ A;  5C7S A;  2ELC A;  4EAF A;  4GIU A;  2WK5 A;  4OWM A;  1ZYK A;  4ZOF A;  4EAD A;  1BRW A;  4N8Q A;  1AZY A;  3TWP A;  4OWU A;  4ZOK A;  4F3F C;  4M0R A;  4OWV A;  2GVQ A;  4N93 A;  5C2L A;  2BPQ A;  1GXB A;  4X5B A;  1ZXY A;  4GA5 A;  4HKM A;  5C1R A;  4YYY A;  4OWO A;  5BO3 A;  3UU1 A;  2DSJ A;  4ZTV A;  5BYT A;  4MUO A;  4GA6 A;  2WK6 A;  4IJ1 A;  4XR5 A;  3QS8 A;  2J0F A;  1V8G A;  1VQU A;  4OWN A;  4GTN A;  1KGZ A;  3QQS A;  3R88 A;  4OWQ A;  4GKM A;  4X5C A;  1RF8 B;  4OWS A;  1KHD A;  1UOU A;  4X5E A;  1OTP A;  3R6C A; 
#chains in the Genus database with same CATH homology
 5BNE A;  4X58 A;  1O17 A;  4YI7 A;  4X46 A;  4LHM A;  4GA4 A;  4YEK A;  4X5D A;  3QR9 A;  1ZVW A;  5EP8 A;  3H5Q A;  3GBR A;  3QSA A;  4X5A A;  2TPT A;  4N5V A;  5BO2 A;  4X59 A;  4ZOJ A;  5EY3 A;  5C7S A;  2ELC A;  4EAF A;  4GIU A;  2WK5 A;  4OWM A;  1ZYK A;  4ZOF A;  4EAD A;  1BRW A;  4N8Q A;  1AZY A;  3TWP A;  4OWU A;  4ZOK A;  4M0R A;  4OWV A;  2GVQ A;  4N93 A;  5C2L A;  2BPQ A;  1GXB A;  4X5B A;  1ZXY A;  4GA5 A;  4HKM A;  5C1R A;  4YYY A;  4OWO A;  5BO3 A;  3UU1 A;  2DSJ A;  4ZTV A;  5BYT A;  4MUO A;  4GA6 A;  2WK6 A;  4IJ1 A;  4XR5 A;  3QS8 A;  2J0F A;  1V8G A;  1VQU A;  4OWN A;  4GTN A;  1KGZ A;  3QQS A;  3R88 A;  4OWQ A;  4GKM A;  4X5C A;  4OWS A;  1KHD A;  1UOU A;  4X5E A;  1OTP A;  3R6C A; 
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