5BO2A

Bianthranilate-like inhibitor with 4-atom "line" and phosphonate "hook" fishing for hydrogen bond donors in mycobacterium tuberculosis anthranilate phosphoribosyltransferase (anprt; trpd)
Total Genus 117
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The genus trace: a function that shows values of genus (vertical axis) for subchains spanned between the first residue, and all other residues (shown on horizontal axis). The number of the latter residue and the genus of a given subchain are shown interactively.

Total Genus
117
sequence length
344
structure length
331
Chain Sequence
SWPQILGRLTDNRDLARGQAAWAMDQIMTGNARPAQIAAFAVAMTMKAPTADEVGELAGVMLSHAHPLPADTVPDDAVDVVGTGTVNLSTMAAIVVAAAGVPVVKHGNRAGADTLEALGVRIDLGPDLVARSLAEVGIGFCFAPRFHPSYRHAAAVRREIGVPTVFNLLGPLTNPARPRAGLIGCAFADLAEVMAGVFAARRSSVLVVHGDDGLDELTTTTTSTIWRVAAGSVDKLTFDPAGFGFARAQLDQLAGGDAQANAAAVRAVLGGARGPVRDAVVLNAAGAIVAHAGLSSEWLPAWEEGLRRASAAIDTGAAEQLLARWVRFGRQ
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The genus matrix. At position (x,y) a genus value for a subchain spanned between x’th and y’th residue is shown. Values of the genus are represented by color, according to the scale given on the right.

Structure visualization

After clicking on a point (x,y) in the genus matrix above, a subchain from x to y is shown in color.

Chord Diagram
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molecule tags Transferase/transferase inhibitor
molecule keywords Anthranilate phosphoribosyltransferase
publication title Binding and mimicking of the phosphate-rich substrate, PRPP.
rcsb
source organism Mycobacterium tuberculosis
total genus 117
structure length 331
sequence length 344
chains with identical sequence B
ec nomenclature ec 2.4.2.18: Anthranilate phosphoribosyltransferase.
pdb deposition date 2015-05-27

pfam database annotations

chain Pfam Accession Code Pfam Family Identifier Pfam Description
A PF00591 Glycos_transf_3 Glycosyl transferase family, a/b domain
A PF02885 Glycos_trans_3N Glycosyl transferase family, helical bundle domain
Image from the rcsb pdb (www.rcsb.org)
cath code
ClassArchitectureTopologyHomologyDomain
1.20.970.10 Mainly Alpha Up-down Bundle Transferase, Pyrimidine Nucleoside Phosphorylase; Chain A, domain 3 Transferase, Pyrimidine Nucleoside Phosphorylase; Chain C 5bo2A01
3.40.1030.10 Alpha Beta 3-Layer(aba) Sandwich Pyrimidine Nucleoside Phosphorylase; Chain A, domain 2 Nucleoside phosphorylase/phosphoribosyltransferase catalytic domain 5bo2A02
2BPQA 4N5VA 1KHDA 4X58A 3R88A 4ZOJA 4N8QA 4ZOKA 1O17A 4GA6A 1OTPA 2TPTA 4X5DA 4YEKA 4YYYA 5BO2A 4OWVA 4X5BA 5EY3A 4LHMA 5C1RA 1ZYKA 4OWUA 5EP8A 2WK6A 1V8GA 4M0RA 4OWMA 4X5CA 4OWOA 4X5AA 4ZOFA 4OWSA 3QR9A 3TWPA 2WK5A 3R6CA 2DSJA 1GXBA 4HKMA 3GBRA 1ZXYA 4YI7A 5BNEA 4ZTVA 4IJ1A 1UOUA 3QQSA 4GA4A 5BO3A 4GIUA 4GKMA 4EAFA 4EADA 3QSAA 4XR5A 4X59A 5C2LA 1KGZA 4GTNA 4MUOA 5BYTA 3H5QA 1VQUA 4X5EA 4GA5A 4OWNA 2GVQA 5C7SA 2ELCA 3QS8A 2J0FA 1AZYA 4N93A 1ZVWA 4X46A 4OWQA 1BRWA 3UU1A
chains in the Genus database with same CATH superfamily
2BPQA 4N5VA 1KHDA 4X58A 3R88A 4ZOJA 4N8QA 4ZOKA 1RRZA 1O17A 4GA6A 1OTPA 2TPTA 4X5DA 4YEKA 4YYYA 5BO2A 4OWVA 4X5BA 5EY3A 4LHMA 5C1RA 1ZYKA 4OWUA 5EP8A 2WK6A 1V8GA 4M0RA 4OWMA 1RF8B 4X5CA 4OWOA 4X5AA 4ZOFA 4OWSA 3QR9A 3TWPA 2WK5A 3R6CA 2DSJA 1GXBA 4HKMA 3GBRA 1ZXYA 4YI7A 5BNEA 4ZTVA 4IJ1A 1UOUA 3QQSA 4GA4A 5BO3A 4GIUA 4GKMA 4EAFA 4EADA 3QSAA 4XR5A 4X59A 5C2LA 4F3FC 1KGZA 4GTNA 4MUOA 5BYTA 3H5QA 1VQUA 4GA5A 4X5EA 4OWNA 2GVQA 5C7SA 2ELCA 3QS8A 2J0FA 1AZYA 4N93A 1ZVWA 4X46A 4OWQA 1BRWA 3UU1A
chains in the Genus database with same CATH topology
2BPQA 4N5VA 1KHDA 4X58A 3R88A 4ZOJA 4N8QA 4ZOKA 1O17A 4GA6A 1OTPA 2TPTA 4X5DA 4YEKA 4YYYA 5BO2A 4OWVA 4X5BA 5EY3A 4LHMA 5C1RA 1ZYKA 4OWUA 5EP8A 2WK6A 1V8GA 4M0RA 4OWMA 4X5CA 4OWOA 4X5AA 4ZOFA 4OWSA 3QR9A 3TWPA 2WK5A 3R6CA 2DSJA 1GXBA 4HKMA 3GBRA 1ZXYA 4YI7A 5BNEA 4ZTVA 4IJ1A 1UOUA 3QQSA 4GA4A 5BO3A 4GIUA 4GKMA 4EAFA 4EADA 3QSAA 4XR5A 4X59A 5C2LA 1KGZA 4GTNA 4MUOA 5BYTA 3H5QA 1VQUA 4X5EA 4GA5A 4OWNA 2GVQA 5C7SA 2ELCA 3QS8A 2J0FA 1AZYA 4N93A 1ZVWA 4X46A 4OWQA 1BRWA 3UU1A
chains in the Genus database with same CATH homology


 
#chains in the Genus database with same CATH superfamily
 2BPQ A;  4N5V A;  1KHD A;  4X58 A;  3R88 A;  4ZOJ A;  4N8Q A;  4ZOK A;  1O17 A;  4GA6 A;  1OTP A;  2TPT A;  4X5D A;  4YEK A;  4YYY A;  5BO2 A;  4OWV A;  4X5B A;  5EY3 A;  4LHM A;  5C1R A;  1ZYK A;  4OWU A;  5EP8 A;  2WK6 A;  1V8G A;  4M0R A;  4OWM A;  4X5C A;  4OWO A;  4X5A A;  4ZOF A;  4OWS A;  3QR9 A;  3TWP A;  2WK5 A;  3R6C A;  2DSJ A;  1GXB A;  4HKM A;  3GBR A;  1ZXY A;  4YI7 A;  5BNE A;  4ZTV A;  4IJ1 A;  1UOU A;  3QQS A;  4GA4 A;  5BO3 A;  4GIU A;  4GKM A;  4EAF A;  4EAD A;  3QSA A;  4XR5 A;  4X59 A;  5C2L A;  1KGZ A;  4GTN A;  4MUO A;  5BYT A;  3H5Q A;  1VQU A;  4X5E A;  4GA5 A;  4OWN A;  2GVQ A;  5C7S A;  2ELC A;  3QS8 A;  2J0F A;  1AZY A;  4N93 A;  1ZVW A;  4X46 A;  4OWQ A;  1BRW A;  3UU1 A; 
#chains in the Genus database with same CATH topology
 2BPQ A;  4N5V A;  1KHD A;  4X58 A;  3R88 A;  4ZOJ A;  4N8Q A;  4ZOK A;  1RRZ A;  1O17 A;  4GA6 A;  1OTP A;  2TPT A;  4X5D A;  4YEK A;  4YYY A;  5BO2 A;  4OWV A;  4X5B A;  5EY3 A;  4LHM A;  5C1R A;  1ZYK A;  4OWU A;  5EP8 A;  2WK6 A;  1V8G A;  4M0R A;  4OWM A;  1RF8 B;  4X5C A;  4OWO A;  4X5A A;  4ZOF A;  4OWS A;  3QR9 A;  3TWP A;  2WK5 A;  3R6C A;  2DSJ A;  1GXB A;  4HKM A;  3GBR A;  1ZXY A;  4YI7 A;  5BNE A;  4ZTV A;  4IJ1 A;  1UOU A;  3QQS A;  4GA4 A;  5BO3 A;  4GIU A;  4GKM A;  4EAF A;  4EAD A;  3QSA A;  4XR5 A;  4X59 A;  5C2L A;  4F3F C;  1KGZ A;  4GTN A;  4MUO A;  5BYT A;  3H5Q A;  1VQU A;  4GA5 A;  4X5E A;  4OWN A;  2GVQ A;  5C7S A;  2ELC A;  3QS8 A;  2J0F A;  1AZY A;  4N93 A;  1ZVW A;  4X46 A;  4OWQ A;  1BRW A;  3UU1 A; 
#chains in the Genus database with same CATH homology
 2BPQ A;  4N5V A;  1KHD A;  4X58 A;  3R88 A;  4ZOJ A;  4N8Q A;  4ZOK A;  1O17 A;  4GA6 A;  1OTP A;  2TPT A;  4X5D A;  4YEK A;  4YYY A;  5BO2 A;  4OWV A;  4X5B A;  5EY3 A;  4LHM A;  5C1R A;  1ZYK A;  4OWU A;  5EP8 A;  2WK6 A;  1V8G A;  4M0R A;  4OWM A;  4X5C A;  4OWO A;  4X5A A;  4ZOF A;  4OWS A;  3QR9 A;  3TWP A;  2WK5 A;  3R6C A;  2DSJ A;  1GXB A;  4HKM A;  3GBR A;  1ZXY A;  4YI7 A;  5BNE A;  4ZTV A;  4IJ1 A;  1UOU A;  3QQS A;  4GA4 A;  5BO3 A;  4GIU A;  4GKM A;  4EAF A;  4EAD A;  3QSA A;  4XR5 A;  4X59 A;  5C2L A;  1KGZ A;  4GTN A;  4MUO A;  5BYT A;  3H5Q A;  1VQU A;  4X5E A;  4GA5 A;  4OWN A;  2GVQ A;  5C7S A;  2ELC A;  3QS8 A;  2J0F A;  1AZY A;  4N93 A;  1ZVW A;  4X46 A;  4OWQ A;  1BRW A;  3UU1 A; 
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