5CGJA

Crystal structure of murine keap1 in complex with ra839, a non-covalent small-molecule binder to keap1 and selective activator of nrf2 signalling.
Total Genus 61
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The genus trace: a function that shows values of genus (vertical axis) for subchains spanned between the first residue, and all other residues (shown on horizontal axis). The number of the latter residue and the genus of a given subchain are shown interactively.

Total Genus
61
sequence length
290
structure length
290
Chain Sequence
VGRLIYTAGGYFRQSLSYLEAYNPSNGSWLRLADLQVPRSGLAGCVVGGLLYAVGGRNNSPDGNTDSSALDCYNPMTNQWSPCASMSVPRNRIGVGVIDGHIYAVGGSHGCIHHSSVERYEPERDEWHLVAPMLTRRIGVGVAVLNRLLYAVGGFDGTNRLNSAECYYPERNEWRMITPMNTIRSGAGVCVLHNCIYAAGGYDGQDQLNSVERYDVETETWTFVAPMRHHRSALGITVHQGKIYVLGGYDGHTFLDSVECYDPDSDTWSEVTRMTSGRSGVGVAVTMEPC
Loading diagram...

The genus matrix. At position (x,y) a genus value for a subchain spanned between x’th and y’th residue is shown. Values of the genus are represented by color, according to the scale given on the right.

Structure visualization

After clicking on a point (x,y) in the genus matrix above, a subchain from x to y is shown in color.

molecule tags Protein binding
molecule keywords Kelch-like ECH-associated protein 1
publication title Characterization of RA839, a Noncovalent Small Molecule Binder to Keap1 and Selective Activator of Nrf2 Signaling.
pubmed doi rcsb
source organism Mus musculus
total genus 61
structure length 290
sequence length 290
ec nomenclature
pdb deposition date 2015-07-09

pfam database annotations

chain Pfam Accession Code Pfam Family Identifier Pfam Description
A PF01344 Kelch_1 Kelch motif
Image from the rcsb pdb (www.rcsb.org)
cath code
ClassArchitectureTopologyHomologyDomain
2.120.10.80 Mainly Beta 6 Propeller Neuraminidase Kelch-type beta propeller 5cgjA00
5FZJA 4IN4A 1X2RA 2DYHA 4ASCA 4L7DA 3VNHA 3ZGDA 2WOZA 2ZWAA 1X2JA 3ADEA 2Z32A 3II7A 2VPJA 4CHBA 2XN4A 4IFNX 5FZNA 3ZGCA 1U6DX 4ZY3A 5CGJA 4IQKA 4XMBA 5FNSA 4IFJA 1ZGKA 3WDZA 3WN7A 4ZGCA 2ZW9A 4CH9A 2FLUX 5FNRA 4IFLX 5FNUA 4L7BA 4N1BA 5FNQA 5FNTA 5F72C 4L7CA 4YY8A 3VNGA 2ZZKA
chains in the Genus database with same CATH superfamily
4IN4A 5GX1A 2DYHA 4MX0A 5D9DA 2VSMA 2VW2A 2RKCA 2HTYA 3P5BL 4FPLA 5D9BA 1F8BA 5H47A 3S2KA 2VWDA 4HW6A 5FZNA 3TIBA 1INVA 4XMBA 1DIMA 1L7FA 4ZLRA 1W8NA 3S94A 1ZGKA 4AHAA 1INHA 2FLUX 4YW4A 4B7JA 4B7QA 1S1DA 4O5SA 4AGTA 1RWLA 1V0FA 2F27A 3S8ZA 6NN9A 4FP2A 4GDJA 4FPYA 4MZEA 1INYA 4MWUA 1X2RA 4MC7A 2HTUA 2AEQA 4YZ4A 3LI4A 1V0ZA 4K3YA 1N1YA 1USXA 1INGA 2XN4A 1IUCA 3H6JA 2F28A 4R40A 4CPLA 4H52A 2H2NA 3G4HA 4NCSA 2F24A 1NCBN 5EX7A 5JYYA 3O4PA 4GN8A 3SLIA 4X49A 2IAVA 1NSBA 5FNQA 4UF7A 4CPNA 1EURA 3WWAA 2CMLA 5FZJA 3TI5A 4UOUA 4XJUA 3NSSA 4C1YB 2YA4A 4Q1UA 4NN9A 4L7DA 2QWJA 3Q6KA 4WA4A 3SRGA 2W20A 1MS3A 5D9CA 3SREA 2OJHA 5FNSA 1Z4VA 4X6KA 1INWA 2VK5A 1INXA 1NCAN 4XOGA 1W1XA 1A4QA 5EO8A 1SLLA 2DSOA 1W20A 1MWEA 2W5NA 2A75A 3TI6A 3PJQA 1B9TA 1NNCA 3TI4A 1CRUA 1B9VA 2SILA 3T1EA 4HZYA 3A9HA 3SOBB 1E1AA 1MR5A 2VSKA 4MWRA 2VPJA 2FHRA 1IJQA 1MS1A 1USRA 1U6DX 5GX5A 2XZIA 2QWBA 3CKZA 2HT8A 2F29A 2G8SA 3H73A 4GEZA 2XZJA 1W8OA 1NN2A 1N6FA 2AEPA 3HLHA 1KITA 1W0OA 4ASCA 2GVUA 3SANA 1SNTA 2BF6A 3K39A 1C9UA 2DG1A 2Z32A 3CL2A 3INBA 2XZKA 3GVKA 4YW1A 1NMCA 5GX4A 1XOEA 3ALWA 5FWWA 4FOWA 4GNAA 4M4NA 4SLIA 3TC9A 4XJZA 4MJUA 3SALA 3LI3A 4QN4A 2C4LA 3DASA 4CPMA 3FVZA 2POOA 4GZOA 5FNUA 1L7GA 1Z50A 3NN9A 4GZPA 4XYXA 2YA7A 4CPOA 3FW0A 4X47A 4XE9A 4L7CA 4D52B 1WP5A 2QWEA 4MWVA 4C1YA 4B7MA 4AGIA 2FP8A 3K38A 3W09A 4K1KA 2VK6A 4FJ6A 2BZDA 3II7A 1Z4YA 2XCYA 1MZ5A 1IVGA 2GVWA 3NO0A 4WA3A 1ZI0A 1NCCN 5HX0A 3TICA 1CRZA 4IYGA 5HUKA 4K1IA 3K36A 3WW9A 2X9MA 3HRPA 4XHXA 2IVZA 1V3CA 3V64C 4XHBA 4MWWA 1V3DA 2IARA 4MJVA 4WEGA 1Z4XA 3Q6TA 4B7RA 4A0PA 2JKBA 1S0JA 5B2DA 1MS4A 4O5TA 4K1HA 1V04A 2HT5A 1IVFA 1IVCA 2F11A 4FPKA 4IFLX 4MWJA 2HTRA 4FOVA 5F9TA 4N1BA 2HQSA 4XJ8A 5M1ZA 3K37A 2QE8A 2V91A 3TIAA 4KS4A 4QN7A 1F8EA 4HZWA 4NC5A 2IATA 2F12A 1EUUA 2BERA 2VVZA 4HHQA 3OPZA 2VK7A 1N6EA 4GN9A 4X4AA 4BBWA 1V3BA 3BYCA 4B7NA 4XIOA 3B69A 4GZTA 1F8CA 2F0ZA 2GHSA 2F26A 2W38A 2QWDA 4YZ2A 4MWYA 1F8DA 1W21A 4M3MA 3A72A 3LI5A 3VNGA 2AH2A 3VNHA 1N7DA 3SOQA 2QWAA 4YW2A 1MS5A 3TI8A 3Q6PA 4YZ5A 2SLIA 1Z4WA 1NNAA 3ADEA 4YZ1A 4XIKA 3BEQA 5NN9A 4ZY3A 5CGJA 2IAOA 2HTWA 1V3EA 1POOA 2FP9A 2HU4A 1NMBN 2QWKA 3HLIA 2ISMA 2W8BB 3CYEA 5GX2A 1SO7A 4YW5A 2YA6A 4HZXA 4H53A 3I1CA 2IAWA 4FPJA 1C5KA 2WOZA 4M4VA 1IVBA 4FPEA 1DILA 3U0SA 5HUNA 4QN3A 4IQKA 1VCUA 3UC1A 4XJQA 2P4OA 4FOQA 3CL0A 4CSDA 2VAQA 3S8VA 1WCQA 1S0IA 3V1SA 4DG6A 4WA5A 2QWIA 1NSDA 2YDPA 3GVJA 2YA5A 1V0EA 2YDTA 2QWFA 3WDZA 4ZGCA 2HTQA 2H2UA 4CH9A 1A14N 1QLGA 3H71A 4FPHA 4FPOB 1E8TA 4D4UA 1VCJA 1WCSA 4GB1A 1IVDA 1QBIA 2F13A 1NNBA 3K3AA 2IASA 3ZGDA 2BATA 4D52C 4CHBA 3GVLA 4MWQA 4KS2A 4Q6KA 4FOYA 4IFJA 4K1JA 2DG0A 2QWCA 3TI3A 3A71A 4XJWA 4FVKA 3E5ZA 2FPBA 2HU0A 5FNTA 1MS9A 5B2CA 4AH4A 3H72A 4KS3A 3O9JA 4J9TA 2W8BA 4MWXA 1N1TA 3SILA 5GTQA 3SOVA 2IAXA 3ALXA 1BJIA 1E8UA 4XILA 1MS0A 1MZ6A 1E8VA 1EUTA 1Z4ZA 2W5OA 3AMSA 4FQ4A 4YZ3A 4IMBA 2VW0A 1SLIA 1NMAN 1PJXA 1S18A 4KS5A 4CPZA 5GX3A 1OFZA 4G3NA 4M4UA 1N1SA 2ZZKA 3G4EA 1CVMA 4D52A 4GNBA 4FP3A 4GZSA 1MS8A 4GZWA 2C4AA 4MZAA 4GZXA 1XOGA 4HZZA 4D8SA 1Q7FA 4I00A 1RWIA 5HUMA 3A9GA 1IUBA 2VW1A 2F25A 1NSCA 2ZW9A 2FPCA 1CQ1A 4QN6A 4GDIA 5FNRA 3V65B 3D12A 4L7BA 4FPFA 4YY8A 4GNCA 3KYAA 4XMIA 4KS1A 1SUUA 3JU4A 1V2IA 2IAPA 4HHOA 7NN9A 2SIMA 4JF7A 2ZB6A 4PWZA 3O9KA 3KGGA 3WN7A 3IAXA 2HT7A 2HTVA 4XJRA 4DGRA 1N1VA 2IAUA 4GJTA 4MWLA 4XJ9A 4HZVA 3L6VA 4GN7A 2ZB5A 2QWGA 1K32A 2B8HA 4GZQA 2IAQA 3AMRA 4QNPA 1N6DA 5EO7A 2QWHA 4QN5A 3DR2A 2ZWAA 4FPCA 1B9SA 1X2JA 4XJAA 2GVVA 4IFNX 1INFA 1IVEA 4JMLA 2YA8A 1EUSA 1L7HA 1W0PA 4XMAA 3ZGCA 3B7EA 1H6LA 1NCDN 4WEFA 2GVXA 4HIZA 4FPGA 3D11A 2F10A 2AGSA 1NPEA 4CPYA 5HUGA 1A4GA 5F72C 4YW3A 4FZHA
chains in the Genus database with same CATH topology
5FZJA 4IN4A 1X2RA 2DYHA 4ASCA 4L7DA 3VNHA 3ZGDA 2WOZA 2ZWAA 1X2JA 3ADEA 2Z32A 3II7A 2VPJA 4CHBA 2XN4A 4IFNX 5FZNA 3ZGCA 1U6DX 4ZY3A 5CGJA 4IQKA 4XMBA 5FNSA 4IFJA 1ZGKA 3WDZA 3WN7A 4ZGCA 2ZW9A 4CH9A 2FLUX 5FNRA 4IFLX 5FNUA 4L7BA 4N1BA 5FNQA 5FNTA 5F72C 4L7CA 4YY8A 3VNGA 2ZZKA
chains in the Genus database with same CATH homology


 
#chains in the Genus database with same CATH superfamily
 5FZJ A;  4IN4 A;  1X2R A;  2DYH A;  4ASC A;  4L7D A;  3VNH A;  3ZGD A;  2WOZ A;  2ZWA A;  1X2J A;  3ADE A;  2Z32 A;  3II7 A;  2VPJ A;  4CHB A;  2XN4 A;  4IFN X;  5FZN A;  3ZGC A;  1U6D X;  4ZY3 A;  5CGJ A;  4IQK A;  4XMB A;  5FNS A;  4IFJ A;  1ZGK A;  3WDZ A;  3WN7 A;  4ZGC A;  2ZW9 A;  4CH9 A;  2FLU X;  5FNR A;  4IFL X;  5FNU A;  4L7B A;  4N1B A;  5FNQ A;  5FNT A;  5F72 C;  4L7C A;  4YY8 A;  3VNG A;  2ZZK A; 
#chains in the Genus database with same CATH topology
 4IN4 A;  5GX1 A;  2DYH A;  4MX0 A;  5D9D A;  2VSM A;  2VW2 A;  2RKC A;  2HTY A;  3P5B L;  4FPL A;  5D9B A;  1F8B A;  5H47 A;  3S2K A;  2VWD A;  4HW6 A;  5FZN A;  3TIB A;  1INV A;  4XMB A;  1DIM A;  1L7F A;  4ZLR A;  1W8N A;  3S94 A;  1ZGK A;  4AHA A;  1INH A;  2FLU X;  4YW4 A;  4B7J A;  4B7Q A;  1S1D A;  4O5S A;  4AGT A;  1RWL A;  1V0F A;  2F27 A;  3S8Z A;  6NN9 A;  4FP2 A;  4GDJ A;  4FPY A;  4MZE A;  1INY A;  4MWU A;  1X2R A;  4MC7 A;  2HTU A;  2AEQ A;  4YZ4 A;  3LI4 A;  1V0Z A;  4K3Y A;  1N1Y A;  1USX A;  1ING A;  2XN4 A;  1IUC A;  3H6J A;  2F28 A;  4R40 A;  4CPL A;  4H52 A;  2H2N A;  3G4H A;  4NCS A;  2F24 A;  1NCB N;  5EX7 A;  5JYY A;  3O4P A;  4GN8 A;  3SLI A;  4X49 A;  2IAV A;  1NSB A;  5FNQ A;  4UF7 A;  4CPN A;  1EUR A;  3WWA A;  2CML A;  5FZJ A;  3TI5 A;  4UOU A;  4XJU A;  3NSS A;  4C1Y B;  2YA4 A;  4Q1U A;  4NN9 A;  4L7D A;  2QWJ A;  3Q6K A;  4WA4 A;  3SRG A;  2W20 A;  1MS3 A;  5D9C A;  3SRE A;  2OJH A;  5FNS A;  1Z4V A;  4X6K A;  1INW A;  2VK5 A;  1INX A;  1NCA N;  4XOG A;  1W1X A;  1A4Q A;  5EO8 A;  1SLL A;  2DSO A;  1W20 A;  1MWE A;  2W5N A;  2A75 A;  3TI6 A;  3PJQ A;  1B9T A;  1NNC A;  3TI4 A;  1CRU A;  1B9V A;  2SIL A;  3T1E A;  4HZY A;  3A9H A;  3SOB B;  1E1A A;  1MR5 A;  2VSK A;  4MWR A;  2VPJ A;  2FHR A;  1IJQ A;  1MS1 A;  1USR A;  1U6D X;  5GX5 A;  2XZI A;  2QWB A;  3CKZ A;  2HT8 A;  2F29 A;  2G8S A;  3H73 A;  4GEZ A;  2XZJ A;  1W8O A;  1NN2 A;  1N6F A;  2AEP A;  3HLH A;  1KIT A;  1W0O A;  4ASC A;  2GVU A;  3SAN A;  1SNT A;  2BF6 A;  3K39 A;  1C9U A;  2DG1 A;  2Z32 A;  3CL2 A;  3INB A;  2XZK A;  3GVK A;  4YW1 A;  1NMC A;  5GX4 A;  1XOE A;  3ALW A;  5FWW A;  4FOW A;  4GNA A;  4M4N A;  4SLI A;  3TC9 A;  4XJZ A;  4MJU A;  3SAL A;  3LI3 A;  4QN4 A;  2C4L A;  3DAS A;  4CPM A;  3FVZ A;  2POO A;  4GZO A;  5FNU A;  1L7G A;  1Z50 A;  3NN9 A;  4GZP A;  4XYX A;  2YA7 A;  4CPO A;  3FW0 A;  4X47 A;  4XE9 A;  4L7C A;  4D52 B;  1WP5 A;  2QWE A;  4MWV A;  4C1Y A;  4B7M A;  4AGI A;  2FP8 A;  3K38 A;  3W09 A;  4K1K A;  2VK6 A;  4FJ6 A;  2BZD A;  3II7 A;  1Z4Y A;  2XCY A;  1MZ5 A;  1IVG A;  2GVW A;  3NO0 A;  4WA3 A;  1ZI0 A;  1NCC N;  5HX0 A;  3TIC A;  1CRZ A;  4IYG A;  5HUK A;  4K1I A;  3K36 A;  3WW9 A;  2X9M A;  3HRP A;  4XHX A;  2IVZ A;  1V3C A;  3V64 C;  4XHB A;  4MWW A;  1V3D A;  2IAR A;  4MJV A;  4WEG A;  1Z4X A;  3Q6T A;  4B7R A;  4A0P A;  2JKB A;  1S0J A;  5B2D A;  1MS4 A;  4O5T A;  4K1H A;  1V04 A;  2HT5 A;  1IVF A;  1IVC A;  2F11 A;  4FPK A;  4IFL X;  4MWJ A;  2HTR A;  4FOV A;  5F9T A;  4N1B A;  2HQS A;  4XJ8 A;  5M1Z A;  3K37 A;  2QE8 A;  2V91 A;  3TIA A;  4KS4 A;  4QN7 A;  1F8E A;  4HZW A;  4NC5 A;  2IAT A;  2F12 A;  1EUU A;  2BER A;  2VVZ A;  4HHQ A;  3OPZ A;  2VK7 A;  1N6E A;  4GN9 A;  4X4A A;  4BBW A;  1V3B A;  3BYC A;  4B7N A;  4XIO A;  3B69 A;  4GZT A;  1F8C A;  2F0Z A;  2GHS A;  2F26 A;  2W38 A;  2QWD A;  4YZ2 A;  4MWY A;  1F8D A;  1W21 A;  4M3M A;  3A72 A;  3LI5 A;  3VNG A;  2AH2 A;  3VNH A;  1N7D A;  3SOQ A;  2QWA A;  4YW2 A;  1MS5 A;  3TI8 A;  3Q6P A;  4YZ5 A;  2SLI A;  1Z4W A;  1NNA A;  3ADE A;  4YZ1 A;  4XIK A;  3BEQ A;  5NN9 A;  4ZY3 A;  5CGJ A;  2IAO A;  2HTW A;  1V3E A;  1POO A;  2FP9 A;  2HU4 A;  1NMB N;  2QWK A;  3HLI A;  2ISM A;  2W8B B;  3CYE A;  5GX2 A;  1SO7 A;  4YW5 A;  2YA6 A;  4HZX A;  4H53 A;  3I1C A;  2IAW A;  4FPJ A;  1C5K A;  2WOZ A;  4M4V A;  1IVB A;  4FPE A;  1DIL A;  3U0S A;  5HUN A;  4QN3 A;  4IQK A;  1VCU A;  3UC1 A;  4XJQ A;  2P4O A;  4FOQ A;  3CL0 A;  4CSD A;  2VAQ A;  3S8V A;  1WCQ A;  1S0I A;  3V1S A;  4DG6 A;  4WA5 A;  2QWI A;  1NSD A;  2YDP A;  3GVJ A;  2YA5 A;  1V0E A;  2YDT A;  2QWF A;  3WDZ A;  4ZGC A;  2HTQ A;  2H2U A;  4CH9 A;  1A14 N;  1QLG A;  3H71 A;  4FPH A;  4FPO B;  1E8T A;  4D4U A;  1VCJ A;  1WCS A;  4GB1 A;  1IVD A;  1QBI A;  2F13 A;  1NNB A;  3K3A A;  2IAS A;  3ZGD A;  2BAT A;  4D52 C;  4CHB A;  3GVL A;  4MWQ A;  4KS2 A;  4Q6K A;  4FOY A;  4IFJ A;  4K1J A;  2DG0 A;  2QWC A;  3TI3 A;  3A71 A;  4XJW A;  4FVK A;  3E5Z A;  2FPB A;  2HU0 A;  5FNT A;  1MS9 A;  5B2C A;  4AH4 A;  3H72 A;  4KS3 A;  3O9J A;  4J9T A;  2W8B A;  4MWX A;  1N1T A;  3SIL A;  5GTQ A;  3SOV A;  2IAX A;  3ALX A;  1BJI A;  1E8U A;  4XIL A;  1MS0 A;  1MZ6 A;  1E8V A;  1EUT A;  1Z4Z A;  2W5O A;  3AMS A;  4FQ4 A;  4YZ3 A;  4IMB A;  2VW0 A;  1SLI A;  1NMA N;  1PJX A;  1S18 A;  4KS5 A;  4CPZ A;  5GX3 A;  1OFZ A;  4G3N A;  4M4U A;  1N1S A;  2ZZK A;  3G4E A;  1CVM A;  4D52 A;  4GNB A;  4FP3 A;  4GZS A;  1MS8 A;  4GZW A;  2C4A A;  4MZA A;  4GZX A;  1XOG A;  4HZZ A;  4D8S A;  1Q7F A;  4I00 A;  1RWI A;  5HUM A;  3A9G A;  1IUB A;  2VW1 A;  2F25 A;  1NSC A;  2ZW9 A;  2FPC A;  1CQ1 A;  4QN6 A;  4GDI A;  5FNR A;  3V65 B;  3D12 A;  4L7B A;  4FPF A;  4YY8 A;  4GNC A;  3KYA A;  4XMI A;  4KS1 A;  1SUU A;  3JU4 A;  1V2I A;  2IAP A;  4HHO A;  7NN9 A;  2SIM A;  4JF7 A;  2ZB6 A;  4PWZ A;  3O9K A;  3KGG A;  3WN7 A;  3IAX A;  2HT7 A;  2HTV A;  4XJR A;  4DGR A;  1N1V A;  2IAU A;  4GJT A;  4MWL A;  4XJ9 A;  4HZV A;  3L6V A;  4GN7 A;  2ZB5 A;  2QWG A;  1K32 A;  2B8H A;  4GZQ A;  2IAQ A;  3AMR A;  4QNP A;  1N6D A;  5EO7 A;  2QWH A;  4QN5 A;  3DR2 A;  2ZWA A;  4FPC A;  1B9S A;  1X2J A;  4XJA A;  2GVV A;  4IFN X;  1INF A;  1IVE A;  4JML A;  2YA8 A;  1EUS A;  1L7H A;  1W0P A;  4XMA A;  3ZGC A;  3B7E A;  1H6L A;  1NCD N;  4WEF A;  2GVX A;  4HIZ A;  4FPG A;  3D11 A;  2F10 A;  2AGS A;  1NPE A;  4CPY A;  5HUG A;  1A4G A;  5F72 C;  4YW3 A;  4FZH A; 
#chains in the Genus database with same CATH homology
 5FZJ A;  4IN4 A;  1X2R A;  2DYH A;  4ASC A;  4L7D A;  3VNH A;  3ZGD A;  2WOZ A;  2ZWA A;  1X2J A;  3ADE A;  2Z32 A;  3II7 A;  2VPJ A;  4CHB A;  2XN4 A;  4IFN X;  5FZN A;  3ZGC A;  1U6D X;  4ZY3 A;  5CGJ A;  4IQK A;  4XMB A;  5FNS A;  4IFJ A;  1ZGK A;  3WDZ A;  3WN7 A;  4ZGC A;  2ZW9 A;  4CH9 A;  2FLU X;  5FNR A;  4IFL X;  5FNU A;  4L7B A;  4N1B A;  5FNQ A;  5FNT A;  5F72 C;  4L7C A;  4YY8 A;  3VNG A;  2ZZK A; 
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similar chains in the Genus database (?% sequence similarity)
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similar chains in the pdb database (?% sequence similarity)

 
#similar chains in the Genus database (?% sequence similarity)
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#similar chains, but unknotted
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#similar chains in the pdb database (?% sequence similarity)
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