236
|
948
|
6xrnA |
Crystal structure of human pi3k-gamma in complex with compound 17 |
310
|
946
|
7jiuA |
Human pi3kdelta in complex with compound 2f |
290
|
1052
|
7mezA |
Structure of the phosphoinositide 3-kinase p110 gamma (pik3cg) p101 (pik3r5) complex |
291
|
925
|
7posA |
Pi3 kinase delta in complex with 5-(3,6-dihydro-2h-pyran-4-yl)-2-methoxy-n-(5-{3-[4-(propan-2-yl)piperazin-1-yl]prop-1-yn-1-yl}pyridin-3-yl)pyridine-3-sulfonamide |
292
|
925
|
7porA |
Pi3 kinase delta in complex with n-[2-(2-fluoro-4-{[4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)pyridin-4-yl]-2-methoxy-5-(morpholin-4-yl)pyridine-3-sulfonamide |
282
|
926
|
7potA |
Pi3 kinase delta in complex with n-[5-(3,6-dihydro-2h-pyran-4-yl)-2-methoxypyridin-3-yl]benzenesulfonamide |
283
|
926
|
7popA |
Pi3 kinase delta in complex with 5-[3,6-dihydro-2h-pyran-4-yl]-2-methoxy-n-[2-methylpyridin-4-yl]pyridine-3-sulfonamide |
275
|
919
|
7oilAAA |
Mpi3kd in complex with compound 58 |
284
|
919
|
7oijAAA |
Mpi3kd in complex with an inhibitor |
286
|
919
|
7oi4AAA |
Mpi3kd in complex with compound 12 |
271
|
919
|
7oisAAA |
Mpi3kd in complex with compound 7 |
255
|
944
|
7jx0A |
Nvs-pi3-4 bound to the pi3kg catalytic subunit p110 gamma |
269
|
947
|
7jwzA |
Ipi-549 bound to the pi3kg catalytic subunit p110 gamma |
270
|
946
|
7jweA |
Gedatolisib bound to the pi3kg catalytic subunit p110 gamma |
290
|
937
|
7k6nA |
Crystal structure of pi3kalpha selective inhibitor 11-1575 |
266
|
937
|
7k6oA |
Crystal structure of pi3kalpha inhibitor 10-5429 |
253
|
936
|
7k71A |
Crystal structure of pi3kalpha inhibitor 4-0686 |
302
|
1013
|
7jisA |
Human pi3kdelta in complex with compound 2f |
282
|
939
|
7k6mA |
Crystal structure of pi3kalpha selective inhibitor pf-06843195 |
295
|
926
|
6zacA |
Pi3k delta in complex with [(dimethylamino)methyldihydrobenzoxazin2methoxypyridinyl]methanesulfonamide |
289
|
926
|
6zaaA |
Pi3k delta in complex with methoxy(methylsulfamoyl)pyridinyln(methylpiperidinyl)dihydrobenzoxazinecarboxamide |
301
|
1012
|
6g6wA |
Human pi3kdelta in complex with ligand lasw1976 |
296
|
926
|
6q73A |
Pi3k delta in complex with n[2chloro5(3,6dihydro2hpyran4yl)pyridin3yl]methanesulfonamide |
296
|
926
|
6q6yA |
Pi3k delta in complex with n(2chloro5phenylpyridin3yl)benzenesulfonamide |
261
|
918
|
6gy0A |
Mpi3kd in complex with az3 |
243
|
942
|
6fh5A |
Pi3kg in complex with compound 7 |
276
|
1084
|
6nctA |
Structure of p110alpha/nish2 - vector data collection |
253
|
919
|
6mulA |
Murine pi3k delta kinsae domain - cpd 1 |
252
|
919
|
6mumA |
Murine pi3k delta kinsae domain - cpd 3 |
325
|
1058
|
5itdA |
Crystal structure of pi3k alpha with pi3k delta inhibitor |
309
|
1052
|
5xgiA |
Crystal structure of pi3k complex with an inhibitor |
295
|
1048
|
5xghA |
Crystal structure of pi3k complex with an inhibitor |
292
|
1048
|
5xgjA |
Crystal structure of pi3k complex with an inhibitor |
287
|
1013
|
5vlrA |
Crystal structure of pi3k delta in complex with a trifluoro-ethyl-pyrazol-pyrolotriazine inhibitor |
298
|
1079
|
5swoA |
Crystal structure of pi3kalpha in complex with fragments 4 and 19 |
281
|
919
|
5ncyA |
Mpi3kd in complex with inh1 |
275
|
919
|
5ngbA |
X-ray diffraction crystal structure of the murine pi3k p110delta in complex with a pan inhibitor |
281
|
916
|
5nczA |
Mpi3kd in complex with inh1 |
275
|
919
|
5t2lA |
Mpi3kd in complex with 7l |
264
|
1011
|
5m6uA |
Human pi3kdelta in complex with lasw1579 |
267
|
925
|
5l72A |
Pi3 kinase delta in complex with n-[6-(5-methanesulfonamido-6-methoxypyridin-3-yl)-1,3-dihydro-2-benzofuran-4-yl]-2-(morpholin-4-yl)acetamide |
251
|
944
|
5jhaA |
Structure of phosphoinositide 3-kinase gamma (pi3k) bound to the potent inhibitor pikin2 |
229
|
948
|
5jhbA |
Structure of phosphoinositide 3-kinase gamma (pi3k) bound to the potent inhibitor pikin3 |
269
|
917
|
5i4uA |
The crystal structure of pi3kdelta with compound 34 |
232
|
918
|
5i6uA |
The crystal structure of pi3kdelta with compound 32 |
340
|
1061
|
5fi4A |
Discovery of imidazo[1,2-a]-pyridine inhibitors of pan-pi3 kinases that are efficacious in a mouse xenograft model |
294
|
1015
|
5dxuA |
P110delta/p85alpha with gdc-0326 |
321
|
1061
|
5dxhA |
P110alpha/p85alpha with compound 5 |
265
|
942
|
5edsA |
Crystal structure of human pi3k-gamma in complex with benzimidazole inhibitor 5 |
258
|
948
|
4urkA |
Pi3kg in complex with azd6482 |