|
35
|
105
|
9kemA |
Crystal structure of brd4-bd1 in complex with h2ak5ack9ac |
|
42
|
126
|
9vczA |
The crystal structure of brd4-bd1 in complex with inhibitor 39b |
|
31
|
105
|
9r5nA |
Fkbp12 in complex with binfunctional ligand b3c and the first bromodomain of brd4 |
|
21
|
107
|
9r5nC |
Fkbp12 in complex with binfunctional ligand b3c and the first bromodomain of brd4 |
|
22
|
107
|
9qw8C |
Fkbp12 in complex with bifunctional ligand 1ad and the first bromodomain of brd4 |
|
40
|
126
|
9qw8A |
Fkbp12 in complex with bifunctional ligand 1ad and the first bromodomain of brd4 |
|
44
|
124
|
9zytAAA |
Crystal structure of brd4 bromodomain bd1 in complex with small molecule plx-3618 |
|
38
|
126
|
9mxkA |
Brd4-bd1 in complex with cyclic peptide 4.1c |
|
1
|
16
|
9mxkB |
Brd4-bd1 in complex with cyclic peptide 4.1c |
|
39
|
125
|
9mpiA |
Brd4-bd1 in complex with cyclic peptide 4.1a |
|
0
|
17
|
9mpiB |
Brd4-bd1 in complex with cyclic peptide 4.1a |
|
0
|
17
|
9mpdC |
Brd4-bd1 in complex with cyclic peptide 4.1b |
|
41
|
109
|
9mpdA |
Brd4-bd1 in complex with cyclic peptide 4.1b |
|
42
|
125
|
9zg4A |
5jc21/cg13250 bound to brd4-bd1. |
|
45
|
127
|
9zg4B |
5jc21/cg13250 bound to brd4-bd1. |
|
23
|
83
|
9vq1A |
Nmr solution structures of brd4 et domain in complex with asxl1 peptide |
|
0
|
14
|
9vq1B |
Nmr solution structures of brd4 et domain in complex with asxl1 peptide |
|
0
|
12
|
9nn5B |
Bet brd4-bd1 in complex with peptide 9.2 |
|
41
|
126
|
9nntA |
Bet brd4-bd1 in complex with peptide 6.1 |
|
0
|
8
|
9nntD |
Bet brd4-bd1 in complex with peptide 6.1 |
|
43
|
126
|
9nn5A |
Bet brd4-bd1 in complex with peptide 9.2 |
|
42
|
126
|
9kt2A |
The crystal structure of bd1 in complex with bds4 |
|
45
|
127
|
9fwxA |
Crystal structure of brd4 bd1 with men1404bs. |
|
44
|
127
|
9fxpA |
Crystal structure of brd4 bd1 with di00626383. |
|
42
|
127
|
9fbyA |
N-terminal bromodomain of human brd4 with (5-(4-chloro-1-((tetrahydro-2h-pyran-4-yl)methyl)-1h-imidazol-2-yl)-1,3-dimethylpyridin-2(1h)-one |
|
44
|
125
|
9f1nA |
First bromodomain of brd4 in complex with isox-dual based degrader 46 |
|
45
|
124
|
9f1jA |
First bromodomain of brd4 in complex with isox-dual based degrader 14 |
|
42
|
124
|
9f1mA |
First bromodomain of brd4 in complex with isox-dual based degrader 45 |
|
43
|
124
|
9f1kA |
First bromodomain of brd4 in complex with isox-dual based inhibitor 30 |
|
43
|
126
|
9f1lA |
First bromodomain of brd4 in complex with isox-dual based degrader 35 |
|
43
|
126
|
8qapA |
Crystal structure of the first bromodomain of brd4 in complex with acetyl-pyrrole derivative compound 2 |
|
43
|
126
|
8qalA |
Crystal structure of the first bromodomain of brd4 in complex with acetyl-pyrrole derivative compound 83 |
|
43
|
126
|
8qarA |
Crystal structure of the first bromodomain of brd4 in complex with acetyl-pyrrole derivative compound 98 |
|
42
|
126
|
8qanA |
Crystal structure of the first bromodomain of brd4 in complex with acetyl-pyrrole derivative compound 79 |
|
24
|
97
|
8ymbC |
The crystal structure of shd931 in complex with brd4-bd2 and vcb |
|
42
|
125
|
8ymhA |
Brd4-bd1 in complex with 5-methyl-2-{[(2r)-2-methyl-4-methylsulfonyl-piperazin-1-yl]methyl}-7-(1-methylpyrazol-3-yl)furo[3,2-c]pyridin-4-one |
|
40
|
126
|
8ymiA |
Brd4-bd1 in complex with 2-{[(3s)-1-benzylpyrrolidin-3-yl]methyl}-5-methyl-7-(1-methylpyrazol-3-yl)pyrazolo[4,3-c]pyridin-4-one |
|
37
|
125
|
8ymfA |
Brd4-bd1 in complex with 7-[2-(cyclopropylmethoxy)phenyl]-5-methyl-2-[(1-methylsulfonyl-4-piperidyl)methyl]pyrazolo[4,3-c]pyridin-4-one |
|
40
|
127
|
8ymeA |
Brd4-bd1 in complex with n-cyclohexyl-1-methyl-6-{[5-methyl-7-(1-methylpyrazol-3-yl)-4-oxo-pyrazolo[4,3-c]pyridin-2-yl]methyl}azepan-1-ium-4-carboxamide 2,2,2-trifluoroacetate |
|
39
|
126
|
8ymgA |
Brd4-bd1 in complex with 7-[4-chloro-1-(tetrahydropyran-4-ylmethyl)imidazol-2-yl]-5-methyl-2-{[(2r)-2-methyl-4-methylsulfonyl-piperazin-1-yl]methyl}furo[3,2-c]pyridin-4-one |
|
39
|
148
|
8ymbD |
The crystal structure of shd931 in complex with brd4-bd2 and vcb |
|
30
|
108
|
8ymbA |
The crystal structure of shd931 in complex with brd4-bd2 and vcb |
|
20
|
104
|
8ymbB |
The crystal structure of shd931 in complex with brd4-bd2 and vcb |
|
44
|
126
|
8v9fA |
Brd4 bd1 liganded with macrocyclic compound 2d (jj-ii-363a) |
|
45
|
127
|
8v92A |
Brd4 bd1 liganded with macrocyclic compound 2b (jj-ii-352a) |
|
44
|
127
|
9qnvA |
Crystal structure of the first bromodomain of human brd4 in complex with compound 2 |
|
43
|
124
|
9qobA |
Crystal structure of the first bromodomain of human brd4 in complex with compound 4 |
|
39
|
123
|
9iv5A |
Brd4 in complex with compound7 |
|
44
|
127
|
9ht2A |
A novel bottom-up approach to find lead-compounds in billion-sized libraries |
|
42
|
127
|
9ht0A |
A novel bottom-up approach to find lead-compounds in billion-sized libraries |
