54
|
164
|
9ax6C |
Tricomplex of rmc-6236, kras g12d, and cypa |
57
|
168
|
9ax6A |
Tricomplex of rmc-6236, kras g12d, and cypa |
65
|
170
|
8t4vA |
Crystal structure of compound 1 bound to k-ras(g12d) |
16
|
76
|
8t74B |
Crystal structure of kras4a (gmppnp) in complex with raf1 (rbd) |
63
|
168
|
8t73A |
Crystal structure of kras4a-r151g with bound gdp and mg ion |
21
|
132
|
8t75B |
Crystal structure of kras4a (gmppnp) in complex with raf1 (rbd-crd) |
52
|
170
|
8t75A |
Crystal structure of kras4a (gmppnp) in complex with raf1 (rbd-crd) |
58
|
170
|
8t71B |
Crystal structure of wt kras4a with bound gdp and mg ion |
58
|
170
|
8t74A |
Crystal structure of kras4a (gmppnp) in complex with raf1 (rbd) |
54
|
169
|
8t72A |
Crystal structure of wt kras4a with bound gmppnp and mg ion |
63
|
171
|
8t71A |
Crystal structure of wt kras4a with bound gdp and mg ion |
59
|
169
|
8tbnA |
Tricomplex of rmc-7977, kras g12s, and cypa |
51
|
164
|
8tbkC |
Tricomplex of rmc-7977, kras g12c, and cypa |
53
|
165
|
8tbnC |
Tricomplex of rmc-7977, kras g12s, and cypa |
54
|
165
|
8tbmC |
Tricomplex of rmc-7977, kras g12v, and cypa |
53
|
165
|
8tbfC |
Tricomplex of rmc-7977, kras wt, and cypa |
52
|
163
|
8tbhC |
Tricomplex of rmc-7977, kras g12r, and cypa |
55
|
165
|
8tbjC |
Tricomplex of rmc-7977, kras g12a, and cypa |
60
|
170
|
8tbjA |
Tricomplex of rmc-7977, kras g12a, and cypa |
61
|
168
|
8tblA |
Tricomplex of rmc-7977, kras g12d, and cypa |
62
|
170
|
8tbkA |
Tricomplex of rmc-7977, kras g12c, and cypa |
60
|
170
|
8tbhA |
Tricomplex of rmc-7977, kras g12r, and cypa |
52
|
165
|
8tblC |
Tricomplex of rmc-7977, kras g12d, and cypa |
60
|
168
|
8tbmA |
Tricomplex of rmc-7977, kras g12v, and cypa |
60
|
170
|
8tbfA |
Tricomplex of rmc-7977, kras wt, and cypa |
67
|
169
|
8jgdA |
Gdp-bound kras g12c in complex with yk-8s |
61
|
168
|
8un3A |
Kras-g13d-gdp in complex with cpd5 (1-((s)-10-(6-amino-4-methyl-3-(trifluoromethyl)pyridin-2-yl)-11-chloro-7-(((2s,4r)-4-fluoro-1-methylpyrrolidin-2-yl)methoxy)-3,4,13,13a-tetrahydropyrazino[2',1':3,4][1,4]oxazepino[5,6,7-de]quinazolin-2(1h)-yl)prop-2-en-1-one) |
62
|
170
|
8un4A |
Kras-g13d-gdp in complex with cpd36 ((e)-1-((3s)-4-(7-(6-amino-4-methyl-3-(trifluoromethyl)pyridin-2-yl)-6-chloro-8-fluoro-2-(((s)-2-methylenetetrahydro-1h-pyrrolizin-7a(5h)-yl)methoxy)quinazolin-4-yl)-3-methylpiperazin-1-yl)-3-(4-((dimethylamino)methyl)-5-methylpyridin-2-yl)prop-2-en-1-one) |
65
|
169
|
8un5A |
Kras-g13d-gdp in complex with cpd38 ((e)-1-((3s)-4-(7-(6-amino-4-methyl-3-(trifluoromethyl)pyridin-2-yl)-6-chloro-8-fluoro-2-(((s)-2-methylenetetrahydro-1h-pyrrolizin-7a(5h)-yl)methoxy)quinazolin-4-yl)-3-methylpiperazin-1-yl)-3-(1,2,3,4-tetrahydroisoquinolin-8-yl)prop-2-en-1-one) |
68
|
169
|
7t47A |
Kras g12d (gppcp) with mrtx-1133 |
57
|
170
|
7rp2A |
Crystal structure of kas g12c in complex with 2h11 clamp |
43
|
215
|
7rp2I |
Crystal structure of kas g12c in complex with 2h11 clamp |
64
|
183
|
7q9uAAA |
Crystal structure of the high affinity kras mutant pde6d complex |
44
|
150
|
7q9uCCC |
Crystal structure of the high affinity kras mutant pde6d complex |
62
|
170
|
6ws2A |
Crystal structure of kras-k104q mutant, gdp-bound |
61
|
169
|
6ws4A |
Crystal structure of kras-g12d/k104q mutant, gdp-bound |
40
|
225
|
7rp2H |
Crystal structure of kas g12c in complex with 2h11 clamp |
68
|
170
|
8qugA |
Kras-g12c in complex with compound 1 |
62
|
176
|
8fmkA |
Crystal structure of human kras with extended switch i loop |
67
|
170
|
8fmjA |
Crystal structure of human kras in space group r32 |
68
|
170
|
7r0nA |
Krasg12c in complex with gdp and compound 2 |
60
|
168
|
7r0qA |
Krasg12c in complex with gdp and compound 3 |
64
|
168
|
7r0mA |
Krasg12c in complex with gdp and jdq443 |
62
|
168
|
7oo7A |
Krasg12c ligand complex |
58
|
169
|
7mquA |
The haddock model of gdp kras in complex with promethazine using nmr chemical shift perturbations |
62
|
168
|
7o70A |
Krasg12c ligand complex |
60
|
170
|
8edyA |
Kras4b a146t 1-185 bound to gdp |
64
|
175
|
8eieA |
Kras4b k117n 1-185 bound to gnp-mg2+ |
62
|
171
|
8ecrA |
Kras4b wt 1-185 bound to gdp-mg2+ |
57
|
169
|
8stmA |
Crystal structure of kras-g75a mutant, gdp-bound |