|
112
|
352
|
3zs5A |
Structural basis for kinase selectivity of three clinical p38alpha inhibitors |
|
94
|
339
|
4ae9A |
Structure and function of the human sperm-specific isoform of protein kinase a (pka) catalytic subunit c alpha 2 |
|
80
|
290
|
4a4oA |
Crystal structure of polo-like kinase 1 in complex with a 2-(2-amino- pyrimidin-4-yl)-1,5,6,7-tetrahydro-pyrrolopyridin-4-one inhibitor |
|
81
|
290
|
4a4lA |
Crystal structure of polo-like kinase 1 in complex with a 5-(2-amino- pyrimidin-4-yl)-1h-pyrrole inhibitor |
|
77
|
284
|
4a07A |
Human pdk1 kinase domain in complex with allosteric activator ps171 bound to the pif-pocket |
|
89
|
317
|
4agdA |
Crystal structure of vegfr2 (juxtamembrane and kinase domains) in complex with sunitinib (su11248) (n-2-diethylaminoethyl)-5-((z)-(5- fluoro-2-oxo-1h-indol-3-ylidene)methyl)-2,4-dimethyl-1h-pyrrole-3- carboxamide) |
|
106
|
347
|
3zsiA |
X-ray structure of p38alpha bound to vx-745 |
|
95
|
350
|
4achA |
Gsk3b in complex with inhibitor |
|
98
|
350
|
4accA |
Gsk3b in complex with inhibitor |
|
104
|
349
|
3zrkA |
Identification of 2-(4-pyridyl)thienopyridinones as gsk-3beta inhibitors |
|
107
|
344
|
3zo2A |
The synthesis and evaluation of diazaspirocyclic protein kinase inhibitors |
|
90
|
282
|
4an2A |
Crystal structures of human mek1 with carboxamide-based allosteric inhibitor xl518 (gdc-0973), or related analogs. |
|
93
|
302
|
4a9sA |
Crystal structure of human chk2 in complex with benzimidazole carboxamide inhibitor |
|
96
|
308
|
4anlA |
Structure of g1269a mutant anaplastic lymphoma kinase |
|
95
|
293
|
3zxzA |
X-ray structure of pf-04217903 bound to the kinase domain of c-met |
|
107
|
358
|
3zyaA |
Human p38 map kinase in complex with 2-amino-phenylamino- dibenzosuberone |
|
111
|
349
|
3zshA |
X-ray structure of p38alpha bound to scio-469 |
|
107
|
349
|
4afjA |
5-aryl-4-carboxamide-1,3-oxazoles: potent and selective gsk-3 inhibitors |
|
107
|
349
|
3zrlA |
Identification of 2-(4-pyridyl)thienopyridinones as gsk-3beta inhibitors |
|
99
|
303
|
4apcA |
Crystal structure of human nima-related kinase 1 (nek1) |
|
96
|
292
|
4appA |
Crystal structure of the human p21-activated kinase 4 in complex with (s)-n-(5-(3-benzyl-1-methylpiperazine-4-carbonyl)-6,6-dimethyl-1,4,5, 6-tetrahydropyrrolo(3,4-c)pyrazol-3-yl)-3-phenoxybenzamide |
|
91
|
304
|
4a9tA |
Crystal structure of human chk2 in complex with benzimidazole carboxamide inhibitor |
|
77
|
277
|
4a4xA |
Nek2-ede bound to cct248662 |
|
87
|
282
|
4an3A |
Crystal structures of human mek1 with carboxamide-based allosteric inhibitor xl518 (gdc-0973), or related analogs. |
|
93
|
286
|
3zzeA |
Crystal structure of c-met kinase domain in complex with n'-((3z)-4- chloro-7-methyl-2-oxo-1,2-dihydro-3h-indol-3-ylidene)-2-(4- hydroxyphenyl)propanohydrazide |
|
113
|
359
|
3zuvA |
Crystal structure of a designed selected ankyrin repeat protein in complex with the phosphorylated map kinase erk2 |
|
104
|
349
|
4a9yA |
P38alpha map kinase bound to cmpd 8 |
|
113
|
328
|
4anmA |
Complex of ck2 with a cdc7 inhibitor |
|
54
|
176
|
4annA |
Crystal structure staphylococcus aureus essb cytoplasmic fragment |
|
77
|
274
|
4aluA |
Benzofuropyrimidinone inhibitors of pim-1 |
|
74
|
269
|
4af3A |
Human aurora b kinase in complex with incenp and vx-680 |
|
89
|
303
|
4a9rA |
Crystal structure of human chk2 in complex with benzimidazole carboxamide inhibitor |
|
87
|
299
|
4aotA |
Crystal structure of human serine threonine kinase-10 (lok) bound to gw830263a |
|
114
|
351
|
4aa4A |
P38alpha map kinase bound to cmpd 22 |
|
91
|
293
|
4aoiA |
Crystal structure of c-met kinase domain in complex with 4-(3-((1h- pyrrolo(2,3-b)pyridin-3-yl)methyl)-(1,2,4)triazolo(4,3-b)(1,2,4) triazin-6-yl)benzonitrile |
|
80
|
273
|
4alwA |
Benzofuropyrimidinone inhibitors of pim-1 |
|
85
|
285
|
3zzwA |
Crystal structure of the kinase domain of ror2 |
|
103
|
312
|
4aseA |
Crystal structure of vegfr2 (juxtamembrane and kinase domains) in complex with tivozanib (av-951) |
|
98
|
312
|
3zosA |
Structure of the ddr1 kinase domain in complex with ponatinib |
|
101
|
350
|
4acdA |
Gsk3b in complex with inhibitor |
|
91
|
293
|
4ap7A |
Crystal structure of c-met kinase domain in complex with 4-((6-(4- fluorophenyl)-(1,2,4)triazolo(4,3-b)(1,2,4)triazin-3-yl)methyl)phenol |
|
68
|
209
|
4anoA |
Crystal structure geobacillus thermodenitrificans essb cytoplasmic fragment |
|
87
|
282
|
4an9A |
Crystal structures of human mek1 with carboxamide-based allosteric inhibitor xl518 (gdc-0973), or related analogs. |
|
89
|
310
|
3zutA |
The structure of ost1 (d160a) kinase |
|
110
|
348
|
4aa5A |
P38alpha map kinase bound to cmpd 33 |
|
96
|
309
|
4ansA |
Structure of l1196m,g1269a double mutant anaplastic lymphoma kinase in complex with crizotinib |
|
109
|
347
|
4aa0A |
P38alpha map kinase bound to cmpd 2 |
|
81
|
274
|
4alvA |
Benzofuropyrimidinone inhibitors of pim-1 |
|
100
|
303
|
4ag8A |
Crystal structure of the vegfr2 kinase domain in complex with axitinib (ag-013736) (n-methyl-2-(3-((e)-2-pyridin-2-yl-vinyl)-1h- indazol-6-ylsulfanyl)-benzamide) |
|
94
|
350
|
4acgA |
Gsk3b in complex with inhibitor |
