|
248
|
1044
|
8ilsA |
Cryo-em structure of pi3kalpha in complex with compound 17 |
|
249
|
1044
|
8ilrA |
Cryo-em structure of pi3kalpha in complex with compound 16 |
|
236
|
1044
|
8ilvA |
Cryo-em structure of pi3kalpha in complex with compound 18 |
|
304
|
1053
|
8sbjA |
Co-structure phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform complexed with brain penetrant inhibitors |
|
284
|
1052
|
8dp0A |
Structure of p110 gamma bound to the ras inhibitory nanobody nb7 |
|
271
|
941
|
8ow2A |
Crystal structure of the p110alpha catalytic subunit from homo sapiens in complex with activator 1938 |
|
299
|
1012
|
8bcyA |
Human pi3kdelta in complex with compound 13 |
|
333
|
1043
|
8aj8A |
Structure of p110 gamma bound to the p84 regulatory subunit |
|
291
|
940
|
8bfuA |
Crystal structure of the apo p110alpha catalytic subunit from homo sapiens |
|
231
|
944
|
8guaA |
Cryo-em structure of cancer-specific pi3kalpha mutant e542k in complex with byl-719 |
|
307
|
1051
|
7tz7A |
Pi3k alpha in complex with an inhibitor |
|
310
|
945
|
8exvA |
Crystal structure of pi3k-alpha in complex with compound 32 |
|
319
|
945
|
8exuA |
Crystal structure of pi3k-alpha in complex with compound 30 |
|
306
|
945
|
8exoA |
Crystal structure of pi3k-alpha in complex with compound 19 |
|
305
|
945
|
8exlA |
Crystal structure of pi3k-alpha in complex with taselisib |
|
288
|
1032
|
8gubA |
Cryo-em structure of cancer-specific pi3kalpha mutant h1047r in complex with byl-719 |
|
206
|
944
|
8gudA |
Cryo-em structure of cancer-specific pi3kalpha mutant e545k in complex with byl-719 |
|
291
|
1034
|
8dcpA |
Pi 3-kinase alpha with nanobody 3-126 |
|
222
|
1031
|
8dcxA |
Pi 3-kinase alpha with nanobody 3-159 |
|
244
|
1041
|
8dd4A |
Pi 3-kinase alpha with nanobody 3-142 |
|
257
|
1046
|
8dd8A |
Pi 3-kinase alpha with nanobody 3-142, crosslinked with dsg |
|
267
|
896
|
7z74A |
Pi3kc2a core in complex with pitcoin2 |
|
250
|
897
|
8a9iA |
Pi3kc2a core in complex with pitcoin1 |
|
358
|
1063
|
7pg5A |
Crystal structure of pi3kalpha |
|
354
|
1063
|
7pg6A |
Crystal structure of pi3kalpha in complex with the inhibitor nvp-byl719 |
|
262
|
897
|
7z75A |
Pi3kc2a core in complex with pitcoin3 |
|
262
|
919
|
7r26A |
Pi3k delta in complex with sd5 |
|
255
|
949
|
7z61A |
Crystal structure of pi3kgamma with a dihydropurinone inhibitor (compound 18) |
|
236
|
948
|
6xrnA |
Crystal structure of human pi3k-gamma in complex with compound 17 |
|
310
|
946
|
7jiuA |
Human pi3kdelta in complex with compound 2f |
|
290
|
1052
|
7mezA |
Structure of the phosphoinositide 3-kinase p110 gamma (pik3cg) p101 (pik3r5) complex |
|
291
|
925
|
7posA |
Pi3 kinase delta in complex with 5-(3,6-dihydro-2h-pyran-4-yl)-2-methoxy-n-(5-{3-[4-(propan-2-yl)piperazin-1-yl]prop-1-yn-1-yl}pyridin-3-yl)pyridine-3-sulfonamide |
|
292
|
925
|
7porA |
Pi3 kinase delta in complex with n-[2-(2-fluoro-4-{[4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)pyridin-4-yl]-2-methoxy-5-(morpholin-4-yl)pyridine-3-sulfonamide |
|
282
|
926
|
7potA |
Pi3 kinase delta in complex with n-[5-(3,6-dihydro-2h-pyran-4-yl)-2-methoxypyridin-3-yl]benzenesulfonamide |
|
283
|
926
|
7popA |
Pi3 kinase delta in complex with 5-[3,6-dihydro-2h-pyran-4-yl]-2-methoxy-n-[2-methylpyridin-4-yl]pyridine-3-sulfonamide |
|
275
|
919
|
7oilAAA |
Mpi3kd in complex with compound 58 |
|
284
|
919
|
7oijAAA |
Mpi3kd in complex with an inhibitor |
|
271
|
919
|
7oisAAA |
Mpi3kd in complex with compound 7 |
|
286
|
919
|
7oi4AAA |
Mpi3kd in complex with compound 12 |
|
255
|
944
|
7jx0A |
Nvs-pi3-4 bound to the pi3kg catalytic subunit p110 gamma |
|
269
|
947
|
7jwzA |
Ipi-549 bound to the pi3kg catalytic subunit p110 gamma |
|
270
|
946
|
7jweA |
Gedatolisib bound to the pi3kg catalytic subunit p110 gamma |
|
290
|
937
|
7k6nA |
Crystal structure of pi3kalpha selective inhibitor 11-1575 |
|
266
|
937
|
7k6oA |
Crystal structure of pi3kalpha inhibitor 10-5429 |
|
253
|
936
|
7k71A |
Crystal structure of pi3kalpha inhibitor 4-0686 |
|
302
|
1013
|
7jisA |
Human pi3kdelta in complex with compound 2f |
|
282
|
939
|
7k6mA |
Crystal structure of pi3kalpha selective inhibitor pf-06843195 |
|
295
|
926
|
6zacA |
Pi3k delta in complex with [(dimethylamino)methyldihydrobenzoxazin2methoxypyridinyl]methanesulfonamide |
|
289
|
926
|
6zaaA |
Pi3k delta in complex with methoxy(methylsulfamoyl)pyridinyln(methylpiperidinyl)dihydrobenzoxazinecarboxamide |
|
301
|
1012
|
6g6wA |
Human pi3kdelta in complex with ligand lasw1976 |