|
39
|
125
|
8p9fA |
Crystal structure of the first bromodomain of human brd4 in complex with the dual bet/hdac inhibitor nb161 |
|
41
|
125
|
8p9lA |
Crystal structure of the first bromodomain of human brd4 in complex with the dual bet/hdac inhibitor nb512 |
|
44
|
127
|
7ugfA |
First bromodomain of brd4 liganded with bms-536924 |
|
44
|
127
|
8e17B |
Brd4-d1 in complex with bet inhibitor |
|
42
|
127
|
8dyrB |
Brd4-d1 in complex with bet inhibitor |
|
45
|
127
|
8e3wB |
Brd4-d1 in complex with bet inhibitor |
|
42
|
149
|
8bdxD |
Ternary complex between vcb, brd4-bd2 and protac 48 |
|
43
|
149
|
8bdtD |
Ternary complex between vcb, brd4-bd2 and protac 51 |
|
31
|
108
|
8bdtA |
Ternary complex between vcb, brd4-bd2 and protac 51 |
|
26
|
97
|
8bdxC |
Ternary complex between vcb, brd4-bd2 and protac 48 |
|
24
|
104
|
8bdtB |
Ternary complex between vcb, brd4-bd2 and protac 51 |
|
23
|
104
|
8bdxB |
Ternary complex between vcb, brd4-bd2 and protac 48 |
|
35
|
109
|
8bdxA |
Ternary complex between vcb, brd4-bd2 and protac 48 |
|
28
|
97
|
8bdtC |
Ternary complex between vcb, brd4-bd2 and protac 51 |
|
45
|
127
|
7r5bA |
Crystal structure of brd4(1) in complex with the inhibitor mpm2 |
|
42
|
124
|
8gq0A |
Crystal structure of brd4 bromodomain 1 (bd1) in complex with stl233497 |
|
41
|
124
|
8gpzA |
Crystal structure of brd4 bromodomain 1 (bd1) in complex with c239-0012 |
|
42
|
123
|
7ymgA |
Crystal structure of brd4 bromodomain 1 (bd1) in complex with 2-({3-ethyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}amino)-3-(1h-indol-3-yl)propan-1-ol |
|
43
|
123
|
7yq9A |
Crystal structure of brd4 bromodomain 1 (bd1) in complex with n-[2-(1h-indol-3-yl)ethyl]-3-(trifluoromethyl)[1,2,4]triazolo[4,3-b]pyridazin-6-amine |
|
39
|
108
|
7uskA |
Brd4-bd2 ligand free |
|
40
|
127
|
8b5bA |
Human brd4 bromdomain 1 in complex with a h4 peptide containing acetyl lysine and apmtri (h4k5ack8apmtri) |
|
39
|
109
|
7usjA |
Brd4-bd2 in complex with sf2523 |
|
43
|
126
|
8b5cA |
Human brd4 bromdomain 1 in complex with a h4 peptide containing apmtri (h4k5/8apmtri) |
|
44
|
126
|
7qdlAAA |
N-terminal bromodomain of human brd4 with i-bet567 |
|
43
|
129
|
7ze7AAA |
Brd4 in complex with fraglite21 |
|
44
|
129
|
7zfnAAA |
Brd4 in complex with fraglite24 |
|
42
|
129
|
7zfyAAA |
Brd4 in complex with peplite-gly |
|
44
|
129
|
7ze6A |
Brd4 in complex with fraglite10 |
|
44
|
129
|
7zfuAAA |
Brd4 in complex with peplite-pro |
|
43
|
129
|
7zg2AAA |
Brd4 in complex with acetyl-lys |
|
42
|
129
|
7zfzAAA |
Brd4 in complex with peplite-val |
|
43
|
129
|
7zfsAAA |
Brd4 in complex with fraglite32 |
|
43
|
129
|
7zefA |
Brd4 in complex with fraglite22 |
|
45
|
129
|
7zg1AAA |
Brd4 in complex with peplite-tyr |
|
42
|
129
|
7zfvA |
Brd4 in complex with peplite-ala |
|
43
|
129
|
7zftAAA |
Brd4 in complex with fraglite33 |
|
45
|
127
|
8eadA |
Crystal structure of the first bromodomain (bd1) of human brd4 in complex with dual brd4-jak2 inhibitor ma9-177 |
|
34
|
116
|
7w3dA |
Crystal structure of brd4 bromodomain 1 (bd1) in complex with n2-(1,2,3-benzotriazol-5-yl)-n3-(dimethylsulfamoyl)-n6-[(2s)-1-methoxypropan-2-yl]pyridine-2,3,6-triamine |
|
44
|
127
|
7t3fA |
Development of brd4 inhibitors as arsenicals antidotes |
|
41
|
127
|
7ruiA |
Bromodomain-containing protein 4 (brd4) bromodomain 1 (bd1) complexed with xr844 |
|
40
|
113
|
7ruhA |
Bromodomain-containing protein 4 (brd4) bromodomain 2 (bd2) complexed with xr844 |
|
42
|
125
|
7utyA |
First bromodomain of brd4 liganded with compound 2c |
|
42
|
125
|
7uznA |
Crystal structure of the first bromodomain of human brd4 in complex with bmt-206059 aka 2-{(3m)-3-(1,4-dimethyl-1h-1,2,3-triazol-5-yl)-8-fluoro-5-[(s)-(oxan-4-yl)(phenyl)methyl]-5h-pyrido[3,2-b]indol-7-yl}propan-2-ol, triply deuterated on the 4-methyl group |
|
42
|
131
|
7v2jA |
Crystal structure of the first bromodomain of human brd4 in complex with the inhibitor 33 |
|
44
|
131
|
7v1uA |
Crystal structure of the first bromodomain of human brd4 in complex with the inhibitor zj12 |
|
41
|
128
|
7wl4A |
Crystal structure of the first bromodomain of human brd4 in complex with the inhibitor slp-50 |
|
33
|
108
|
7wjsA |
Crystal structure of the first bromodomain of human brd4 in complex with the inhibitor y13157 |
|
34
|
109
|
7wkyA |
Crystal structure of the first bromodomain of human brd4 in complex with the inhibitor y13153 |
|
44
|
126
|
7rjrA |
Crystal structure of human bromodomain containing protein 4 (brd4) in complex with bcltf1 |
|
44
|
127
|
7rmdA |
Crystal structure of the first bromodomain of human brd4 in complex with sj001011461-1 |
