|
43
|
128
|
7khhD |
Ternary complex of vhl/brd4-bd1/compound9 (4-(3,5-difluoropyridin-2-yl)-n-(11-(((s)-1-((2s,4r)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)amino)-11-oxoundecyl)-10-methyl-7-((methylsulfonyl)methyl)-11-oxo-3,4,10,11-tetrahydro-1h-1,4,10-triazadibenzo[cd,f]azulene-6-carboxamide) |
|
44
|
126
|
7khlA |
Brd4-bd1 compound6 (methyl 4-(3,5-difluoropyridin-2-yl)-10-methyl-7-((methylsulfonyl)methyl)-11-oxo-3,4,10,11-tetrahydro-1h-1,4,10-triazadibenzo[cd,f]azulene-6-carboxylate) |
|
45
|
124
|
7bboAAA |
Crystal structure of the second bromodomain of pleckstrin homology domain interacting protein (phip) in space group p212121 |
|
45
|
119
|
5s92A |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
44
|
119
|
5s9eA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
41
|
119
|
5s9hA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
47
|
119
|
5s96A |
Pandda analysis group deposition -- crystal structure of phip in complex with starting material |
|
43
|
119
|
5s9cA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
43
|
119
|
5s8rA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
43
|
119
|
5s8tA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
43
|
119
|
5s8uA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
46
|
119
|
5s8xA |
Pandda analysis group deposition -- crystal structure of phip in complex with starting material |
|
45
|
119
|
5s9fA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
46
|
119
|
5s9jA |
Pandda analysis group deposition -- crystal structure of phip in complex with starting material |
|
44
|
119
|
5s95A |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
46
|
119
|
5s99A |
Pandda analysis group deposition -- crystal structure of phip in complex with starting material |
|
45
|
119
|
5s8zA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
44
|
119
|
5s94A |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
45
|
119
|
5s9dA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
46
|
119
|
5s8wA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
45
|
119
|
5s8vA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
45
|
119
|
5s9aA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
48
|
119
|
5s91A |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
44
|
119
|
5s8yA |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
44
|
119
|
5s93A |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
44
|
119
|
5s97A |
Pandda analysis group deposition -- crystal structure of phip in complex with z198194396 synthetic derivative |
|
42
|
113
|
6zb2AAA |
C-terminal bromodomain of human brd2 with gsk549 |
|
44
|
115
|
6zb0AAA |
C-terminal bromodomain of human brd2 with 1-benzyl-n-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide |
|
44
|
127
|
6zb3AAA |
N-terminal bromodomain of human brd4 with gsk620 |
|
42
|
112
|
6zb1AAA |
C-terminal bromodomain of human brd2 with gsk620 |
|
42
|
127
|
6x7cA |
Brd4 bromodomain 1 in complex with multi-action inhibitor srx3212 |
|
37
|
124
|
6x7dA |
Brd4 bromodomain 1 in complex with multi-action inhibitor sf2523p |
|
43
|
134
|
6x7bA |
Brd4 bromodomain 1 in complex with multi-action inhibitor srx3212p |
|
44
|
127
|
6sajA |
Crystal structure of brd4(1) bound to inhibitor bux6 (12) |
|
41
|
124
|
6lg5A |
Crystal structure of the first bromodomain of human brd4 in complex with compound bdf-1038 |
|
43
|
124
|
6limA |
Brd4-bd1 bound with compound 40 |
|
42
|
124
|
6lihA |
Brd4 bd1 bound with compound 10 |
|
44
|
124
|
6lg7A |
Crystal structure of the first bromodomain of human brd4 in complex with compound bdf-2030 |
|
42
|
124
|
6lg4A |
Crystal structure of the first bromodomain of human brd4 in complex with compound bdf-1024 |
|
42
|
124
|
6lg6A |
Crystal structure of the first bromodomain of human brd4 in complex with compound bdf-1021 |
|
44
|
119
|
5s8iA |
Xchem group deposition -- crystal structure of the second bromodomain of pleckstrin homology domain interacting protein (phip) in complex with n01186d (space group c2) |
|
42
|
124
|
6lg8A |
Crystal structure of the first bromodomain of human brd4 in complex with compound bdf-2138 |
|
45
|
119
|
5s8lA |
Xchem group deposition -- crystal structure of the second bromodomain of pleckstrin homology domain interacting protein (phip) in complex with e11289c (space group c2) |
|
44
|
120
|
5s8pA |
Xchem group deposition -- crystal structure of the second bromodomain of pleckstrin homology domain interacting protein (phip) in complex with e07179c (space group p212121) |
|
44
|
119
|
5s8dA |
Xchem group deposition -- crystal structure of the second bromodomain of pleckstrin homology domain interacting protein (phip) in complex with n00539e (space group c2) |
|
45
|
119
|
5s8mA |
Xchem group deposition -- crystal structure of the second bromodomain of pleckstrin homology domain interacting protein (phip) in complex with n11511a (space group c2) |
|
45
|
127
|
7a9uAAA |
N-terminal bromodomain of human brd4 with 3-(3-(but-3-yn-1-yl)-3h-diazirin-3-yl)-n-(3-methyl-[1,2,4]triazolo[4,3-a]pyridin-8-yl)propanamide |
|
45
|
117
|
7k6sA |
Crystal structure of the bromodomain (bd) of human bromodomain and phd finger-containing transcription factor (bptf) bound to compound 4 (skt1174) |
|
47
|
124
|
7av9AAA |
Crystal structure of the second bromodomain of pleckstrin homology domain interacting protein (phip) in space group c2 |
|
40
|
105
|
7kdzA |
Crystal structure of the bromodomain (bd) of human bromodomain and phd finger-containing transcription factor (bptf) bound to tp-238 |
