|
65
|
199
|
4pnsA |
Crystal structure of human tankyrase 2 in complex with inh2bp. |
|
61
|
211
|
4n4vA |
Co-crystal structure of tankyrase 1 with compound 4 [(4s)-3-{trans-4-[6-amino-5-(pyrimidin-2-yl)pyridin-3-yl]cyclohexyl}-5,5-dimethyl-4-phenyl-1,3-oxazolidin-2-one] |
|
61
|
212
|
4n4tA |
Co-crystal structure of tankyrase 1 with compound 3 [(4s)-3-{4-[6-amino-5-(pyrimidin-2-yl)pyridin-3-yl]phenyl}-5,5-dimethyl-4-phenyl-1,3-oxazolidin-2-one] |
|
64
|
212
|
4n3rA |
Co-crystal structure of tankyrase 1 with compound 2 (5-(2-aminoquinazolin-6-yl)-n-(4,4-dimethyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)-2-fluorobenzamide) |
|
64
|
211
|
4oa7A |
Crystal structure of tankyrase1 in complex with iwr1 |
|
63
|
211
|
4msgA |
Crystal structure of tankyrase 1 with compound 22 |
|
59
|
211
|
4mskA |
Co-crystal structure of tankyrase 1 with compound 34 |
|
65
|
210
|
4mt9A |
Co-crystal structure of tankyrase 1 with compound 49 |
|
66
|
210
|
4m7bA |
Human tankyrase 2 - catalytic parp domain in complex with an inhibitor upf1854 |
|
67
|
210
|
4li6A |
Tankyrase-1 complexed with small molecule inhibitor n-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-3-phenyl-n-(thiophen-2-ylmethyl)propanamide |
|
46
|
161
|
4l0tA |
Tankyrase 2 in complex with 4'-nitro flavone |
|
44
|
161
|
4kzqA |
Crystal structure of human tankyrase 2 in complex with 4' -hydroxy flavone |
|
104
|
356
|
4l7rA |
Human artd3 (parp3) - catalytic domain in complex with inhibitor me0400 |
|
47
|
161
|
4l09A |
Crystal structure of human tankyrase 2 in complex with 4-(4-oxo-4h-chromen-2-yl)benzoic acid |
|
115
|
357
|
4l6zA |
Human artd3 (parp3) - catalytic domain in complex with inhibitor sto1168 |
|
65
|
209
|
4li8A |
Tankyrase-1 complexed with small molecule inhibitor 2-[4-(4-fluorobenzoyl)piperidin-1-yl]-n-[(4-oxo-3,5,7,8-tetrahydro-4h-pyrano[4,3-d]pyrimidin-2-yl)methyl]-n-(thiophen-2-ylmethyl)acetamide |
|
110
|
356
|
4l7pA |
Human artd3 (parp3) - catalytic domain in complex with inhibitor me0395 |
|
111
|
357
|
4l7oA |
Human artd3 (parp3) - catalytic domain in complex with inhibitor sto1542 |
|
47
|
161
|
4l0sA |
Tankyrase 2 in complex with 4'-cyano flavone |
|
47
|
161
|
4l0vA |
Tankyrase 2 in complex with 4'-chloro flavone |
|
113
|
356
|
4l7nA |
Human artd3 (parp3) - catalytic domain in complex with inhibitor sto1542 |
|
45
|
161
|
4l2fA |
Tankyrase 2 in complex with 6-chloro flavone |
|
45
|
161
|
4l31A |
Tankyrase 2 in complex with methyl 4-(4-oxochromen-2-yl)benzoate |
|
61
|
210
|
4krsA |
Tankyrase-1 complexed with small molecule inhibitor |
|
113
|
357
|
4l70A |
Human artd3 (parp3) - catalytic domain in complex with inhibitor me0352 |
|
110
|
352
|
4l6sA |
Parp complexed with benzo[1,4]oxazin-3-one inhibitor |
|
46
|
161
|
4l2kA |
Tankyrase 2 in complex with 2-(1,3-benzodioxol-5-yl)-4h-chromen-4-one |
|
65
|
211
|
4li7A |
Tankyrase-1 complexed with small molecule inhibitor 4-chloro-5-cyano-n-{2-[4-(4-fluorobenzoyl)piperidin-1-yl]ethyl}-2-methoxybenzamide |
|
110
|
356
|
4l7lA |
Human artd3 (parp3) - catalytic domain in complex with inhibitor me0368 |
|
49
|
161
|
4l10A |
Tankyrase 2 in complex with 4'-methoxy flavone |
|
48
|
161
|
4l0iA |
Tankyrase 2 catalytic domain in complex with ethyl 4-(4-oxo-4h-chromen-2-yl)benzoate |
|
59
|
212
|
4k4fA |
Co-crystal structure of tnks1 with compound 18 [4-[(4s)-5,5-dimethyl-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-n-(quinolin-8-yl)benzamide] |
|
45
|
161
|
4kzuA |
Crystal structure of human tankyrase 2 in complex with 4' -bromo flavone |
|
48
|
161
|
4l32A |
Tankyrase 2 in complex with 2-[4-(4-methylpiperazine-1-carbonyl)phenyl]chromen-4-one |
|
46
|
161
|
4l34A |
Tankyrase 2 in complex with 4'-tetrazole flavone |
|
47
|
161
|
4kzlA |
Crystal structure of human tankyrase 2 in complex with 4'-fluoro flavone |
|
48
|
161
|
4l0bA |
Tankyrase 2 in complex with 4'-dimethylamino flavone |
|
48
|
161
|
4l33A |
Tankyrase 2 in complex with cyanomethyl 4-(4-oxo-4h-chromen-2-yl)benzoate |
|
59
|
212
|
4k4eA |
Co-crystal structure of tnks1 with compound 52 [n~2-(5-chloro-2-methoxyphenyl)-n-[trans-4-(2-oxo-2,3-dihydro-1h-benzimidazol-1-yl)cyclohexyl]glycinamide] |
|
97
|
355
|
4l7uA |
Human artd3 (parp3) - catalytic domain in complex with inhibitor me0398 |
|
45
|
161
|
4l2gA |
Tankyrase 2 in complex with 6- fluoro flavone |
|
59
|
227
|
4hyfA |
Structural basis and sar for od 270, a lead stage 1,2,4-triazole based specific tankyrase1/2 inhibitor |
|
70
|
210
|
4j22A |
Tankyrase 2 in complex with 3-chloro-4-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)-n-[2-(morpholin-4-yl)ethyl]benzamide |
|
70
|
210
|
4j3mA |
Tankyrase 2 in complex with 3-chloro-4-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)benzoic acid |
|
71
|
210
|
4j21A |
Tankyrase 2 in complex with 7-(4-amino-2-chlorophenyl)-4-methylquinolin-2(1h)-one |
|
71
|
210
|
4j3lA |
Tankyrase 2 in complex with 3-chloro-n-(2-methoxyethyl)-4-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)benzamide |
|
69
|
210
|
4j1zA |
Tankyrase 2 in complex with 4-chloro-1,2-dihydrophatalzin-one |
|
68
|
210
|
4iueA |
Tankyrase in complex with 7-(2-fluorophenyl)-4-methyl-1,2-dihydroquinolin-2-one |
|
60
|
212
|
4i9iA |
Crystal structure of tankyrase 1 with compound 4 |
|
46
|
161
|
4hmhA |
Crystal structure of tankyrase 2 in complex with 7,3-dihydroxyflavone |
