|
95
|
246
|
5g46A |
Ligand complex of rorg lbd |
|
92
|
250
|
5gicA |
Crystal structure of vdr in complex with dlam-2p |
|
95
|
244
|
5g45A |
Ligand complex of rorg lbd |
|
98
|
248
|
5g3jA |
Discovery of new selective glucocorticoid receptor agonist leads |
|
100
|
255
|
5gt4A |
Crystal structure of the human vitamin d receptor ligand binding domain complexed with (1r,2s,3r,5z,7e,14beta,17alpha)-2-cyanopropoxy-9,10-secocholesta-5,7,10-triene-1,3,25-triol |
|
99
|
252
|
5g42A |
Ligand complex of rorg lbd |
|
87
|
251
|
5awkA |
Crystal structure of vdr-lbd/partial agonist complex: 22s-ethyl analogue |
|
95
|
271
|
5azvA |
Crystal structure of hppargamma ligand binding domain complexed with 17-oxodha |
|
97
|
245
|
5g44A |
Ligand complex of rorg lbd |
|
95
|
251
|
5awjA |
Crystal structure of vdr-lbd/partial agonist complex: 22s-hexyl analogue |
|
85
|
242
|
5fqpA |
Selective estrogen receptor downregulator antagonists: tetrahydroisoquinoline phenols 1. |
|
84
|
239
|
5fqvA |
Selective estrogen receptor downregulator antagonists: tetrahydroisoquinoline phenols 5. |
|
84
|
239
|
5fqtA |
Selective estrogen receptor downregulator antagonists: tetrahydroisoquinoline phenols 4. |
|
82
|
244
|
5avlA |
Crystal structure of lxralpha in complex with tert-butyl benzoate analog, compound 32b |
|
83
|
239
|
5fqsA |
Selective estrogen receptor downregulator antagonists: tetrahydroisoquinoline phenols 3. |
|
92
|
268
|
5f9bA |
X-ray crystal structure of ppargamma in the complex with caulophyllogenin |
|
84
|
239
|
5fqrA |
Selective estrogen receptor downregulator antagonists: tetrahydroisoquinoline phenols 2. |
|
74
|
243
|
5aviA |
Crystal structure of lxralpha in complex with tert-butyl benzoate analog, compound 4 |
|
87
|
245
|
5eitA |
Crystal structure of the er-alpha ligand-binding domain (y537s) in complex with the imidazopyridine derivative 2-(4-hydroxyphenyl)-3-(trifluoromethyl)imidazo[1,2-a]pyridin-6-ol |
|
79
|
245
|
5egvA |
Crystal structure of the er-alpha ligand-binding domain (y537s) in complex the 3,4-diaryl-furan derivative 3-chloranyl-4-[4-(2-chloranyl-4-oxidanyl-phenyl)furan-3-yl]phenol |
|
101
|
299
|
5e7vA |
Potent vitamin d receptor agonist |
|
94
|
246
|
5e1cA |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative dimethyl {(1s)-3-[bis(4-hydroxyphenyl)methylidene]cyclohexyl}propanedioate |
|
87
|
244
|
5du5A |
Crystal structure of the er-alpha ligand-binding domain in complex with a dichloro-substituted, 3,4-diarylthiophene dioxide core ligand |
|
91
|
243
|
5ei1A |
Crystal structure of the er-alpha ligand-binding domain (y537s) in complex with the imidazopyridine derivative 2-(4-hydroxyphenyl)-3-iodanyl-imidazo[1,2-a]pyridin-6-ol |
|
85
|
210
|
5ec9A |
Retinoic acid receptor alpha in complex with chiral dihydrobenzofuran benzoic acid 9a and a fragment of the coactivator tif2 |
|
87
|
241
|
5dxeA |
Estrogen receptor alpha ligand binding domain y537s mutant in complex with stapled peptide src2-p4 and estradiol |
|
82
|
246
|
5e15A |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative 4,4'-{[4-(2-hydroxyethyl)cyclohexylidene]methanediyl}diphenol |
|
95
|
245
|
5ejvA |
Rory in complex with t090131718 and coactivator peptide ebi96 |
|
99
|
252
|
5aphA |
Ligand complex of rorg lbd |
|
86
|
245
|
5dy8A |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative 4,4'-{[(3s)-3-ethylcyclohexylidene]methanediyl}diphenol |
|
73
|
239
|
5dvvA |
Crystal structure of the er-alpha ligand-binding domain in complex with a triaryl-imine analog 4,4'-(phenylcarbonimidoyl)diphenol |
|
86
|
244
|
5e0xA |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative 4,4'-{[(3s)-3-(4-methoxyphenyl)cyclohexylidene]methanediyl}diphenol |
|
83
|
218
|
5ethA |
Rory in complex with inverse agonist 3. |
|
83
|
244
|
5ehjA |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative 4,4'-[(4ar,8ar)-octahydronaphthalen-2(1h)-ylidenemethanediyl]diphenol |
|
85
|
244
|
5e0wA |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative 4,4'-{[(3s)-3-(4-hydroxyphenyl)cyclohexylidene]methanediyl}diphenol |
|
93
|
242
|
5dxbA |
Estrogen receptor alpha ligand binding domain y537s mutant in complex with stapled peptide src2-p1 and estradiol |
|
88
|
244
|
5e14A |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative 4,4'-{[(3r)-3-phenylcyclohexylidene]methanediyl}diphenol |
|
89
|
229
|
5apkA |
Ligand complex of rorg lbd |
|
101
|
250
|
5apjA |
Ligand complex of rorg lbd |
|
86
|
242
|
5dxgA |
Estrogen receptor alpha ligand binding domain y537s mutant in complex with stapled peptide src2-p5 |
|
86
|
244
|
5e19A |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative methyl {4-[bis(4-hydroxyphenyl)methylidene]cyclohexyl}acetate |
|
91
|
245
|
5dziA |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative 4,4'-{[(3s)-3-(2-hydroxyethyl)cyclohexylidene]methanediyl}diphenol |
|
84
|
246
|
5dzhA |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative 4,4'-{[4-(2-hydroxyethyl)cyclohexylidene]methanediyl}diphenol |
|
81
|
243
|
5dxqA |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative 4,4'-[(1s,5s)-bicyclo[3.3.1]non-9-ylidenemethanediyl]diphenol |
|
89
|
241
|
5dx3A |
Estrogen receptor alpha ligand binding domain y537s mutant in complex with stapled peptide src2-p3 and estradiol |
|
85
|
244
|
5dwiA |
Crystal structure of the er-alpha ligand-binding domain in complex with a resorcinyl 2-chloro-substituted diaryl-imine analog 4-[(e)-[(2-chlorophenyl)imino](4-hydroxyphenyl)methyl]benzene-1,3-diol |
|
87
|
244
|
5drjA |
Crystal structure of the er-alpha ligand-binding domain in complex with a dichloro-substituted, 3-methyl 2,5-diarylthiophene-core ligand 4,4'-(3-methylthiene-2,5-diyl)bis(3-chlorophenol) |
|
86
|
245
|
5dz3A |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative 4,4'-{[4-(fluoromethyl)cyclohexylidene]methanediyl}diphenol |
|
79
|
243
|
5dydA |
Crystal structure of the er-alpha ligand-binding domain in complex with the cyclofenil derivative 4,4'-{[(3s)-3-(methylsulfanyl)cyclohexylidene]methanediyl}diphenol |
|
88
|
248
|
5dweA |
Crystal structure of the er-alpha ligand-binding domain in complex with a 2-chloro-substituted triaryl-imine analog 4,4'-[(2-chlorophenyl)carbonimidoyl]diphenol |
