|
42
|
124
|
6lihA |
Brd4 bd1 bound with compound 10 |
|
42
|
124
|
6lg4A |
Crystal structure of the first bromodomain of human brd4 in complex with compound bdf-1024 |
|
42
|
124
|
6lg6A |
Crystal structure of the first bromodomain of human brd4 in complex with compound bdf-1021 |
|
42
|
124
|
6lg8A |
Crystal structure of the first bromodomain of human brd4 in complex with compound bdf-2138 |
|
45
|
127
|
7a9uAAA |
N-terminal bromodomain of human brd4 with 3-(3-(but-3-yn-1-yl)-3h-diazirin-3-yl)-n-(3-methyl-[1,2,4]triazolo[4,3-a]pyridin-8-yl)propanamide |
|
44
|
127
|
7ajnA |
Crystal structure of the first bromodomain of brd4 in complex with a bzd ligand |
|
45
|
127
|
6rwjA |
Crystal structure of brd4(1) bound to inhibitor bug0 (6) |
|
1
|
14
|
6ulvE |
Brd4-bd1 in complex with the cyclic peptide 4.2_1 |
|
37
|
109
|
6sa3A |
Crystal structure of brd4(1) bound to inhibitor bux4 (13) |
|
44
|
127
|
6s6kA |
Crystal structure of brd4(1) bound to inhibitor bux2 (9) |
|
36
|
108
|
6ulvA |
Brd4-bd1 in complex with the cyclic peptide 4.2_1 |
|
40
|
124
|
6lg9A |
Crystal structure of the first bromodomain of human brd4 in complex with compound bdf-2143 |
|
42
|
127
|
6sb8A |
Crystal structure of brd4(1) bound to inhibitor bux14 (7) |
|
45
|
127
|
6s4bA |
Crystal structure of brd4(1) bound to inhibitor bux1 (8) |
|
43
|
126
|
6zciA |
Crystal structure of brd4-bd1 in complex with nvs-bet-1 |
|
43
|
127
|
6sahA |
Crystal structure of brd4(1) bound to inhibitor bux5 (11) |
|
44
|
127
|
6sa2A |
Crystal structure of brd4(1) bound to inhibitor bux3 (10) |
|
38
|
125
|
6wgxA |
Cocrystal of brd4(d1) with a selective inhibitor |
|
39
|
131
|
6ww8A |
Brd4 bromodomain 1 in complex with triple cdk4/6-pi3k-bet inhibitor |
|
42
|
127
|
6u72A |
Brd4-bd1 in complex with the cyclic peptide 3.1_2_ack5toa |
|
0
|
14
|
6u8gE |
Brd4-bd2 in complex with the cyclic peptide 3.1_2_ack7toa |
|
0
|
14
|
6u6lB |
Brd4-bd2 in complex with the cyclic peptide 3.1_2 |
|
0
|
14
|
6u74E |
Brd4-bd1 in complex with the cyclic peptide 3.1_2 |
|
0
|
17
|
6u8mC |
Brd4-bd1 in complex with the cyclic peptide 3.2_1 |
|
1
|
12
|
6u8iB |
Brd4-bd2 in complex with the cyclic peptide 3.2_2 |
|
35
|
112
|
6u6lA |
Brd4-bd2 in complex with the cyclic peptide 3.1_2 |
|
44
|
126
|
6u0dA |
Crystal structure of the first bromodomain of human brd4 in complex with the inhibitor zl0590 |
|
39
|
125
|
6u8mA |
Brd4-bd1 in complex with the cyclic peptide 3.2_1 |
|
0
|
11
|
6u6kC |
Brd4-bd1 in complex with the cyclic peptide 3.1_3 |
|
0
|
14
|
6u72C |
Brd4-bd1 in complex with the cyclic peptide 3.1_2_ack5toa |
|
39
|
126
|
6u8gA |
Brd4-bd2 in complex with the cyclic peptide 3.1_2_ack7toa |
|
43
|
126
|
6u6kA |
Brd4-bd1 in complex with the cyclic peptide 3.1_3 |
|
0
|
10
|
6ulsB |
Brd4-bd1 in complex with the a diacetylated-e2f1 peptide |
|
42
|
124
|
6ulsA |
Brd4-bd1 in complex with the a diacetylated-e2f1 peptide |
|
38
|
109
|
6u8iA |
Brd4-bd2 in complex with the cyclic peptide 3.2_2 |
|
42
|
128
|
6u74A |
Brd4-bd1 in complex with the cyclic peptide 3.1_2 |
|
38
|
107
|
6ko2A |
Crystal structure of brd4-brmo2 in complex with h2a.zk4ack7ac peptide |
|
41
|
127
|
6keeA |
Crystal structure of brd4 bromodomain1 with an inhibitor |
|
42
|
123
|
6kekA |
Crystal structure of brd4 bromodomain 1 (bd1) in complex with 6-hydroxy-16-methoxy-11-methyl-2-oxa-11-azatetracyclo[8.6.1.03,8.013,17]heptadeca-1(16),3,5,7,9,13(17),14-heptaen-12-one |
|
42
|
123
|
6kejA |
Crystal structure of brd4 bromodomain 1 (bd1) in complex with 6-[2-(diethylamino)ethoxy]-16-methoxy-11-methyl-2-oxa-11-azatetracyclo[8.6.1.03,8.013,17]heptadeca-1(17),3,5,7,9,13,15-heptaen-12-one |
|
43
|
127
|
6kegA |
Brd4 bromodomain1 with an inhibitor |
|
42
|
123
|
6kehA |
Crystal structure of brd4 bromodomain 1 (bd1) in complex with 6,16-dimethoxy-11-methyl-2-oxa-11-azatetracyclo[8.6.1.03,8.013,17]heptadeca-1(17),3,5,7,9,13,15-heptaen-12-one |
|
43
|
123
|
6kecA |
Crystal structure of brd4 bromodomain 1 (bd1) in complex with 4-ethoxy-5,16-dimethoxy-11-methyl-2-oxa-11-azatetracyclo[8.6.1.03,8.013,17]heptadeca-1(17),3,5,7,9,13,15-heptaen-12-one |
|
44
|
127
|
6kefA |
Brd4 bromodomain1 with an inhibitor |
|
43
|
127
|
6kedA |
Brd4 bromodomain1 with an inhibitor |
|
43
|
123
|
6keiA |
Crystal structure of brd4 bromodomain 1 (bd1) in complex with 16-methoxy-11-methyl-6-[(pyridin-2-yl)methoxy]-2-oxa-11-azatetracyclo[8.6.1.03,8.013,17]heptadeca-1(16),3,5,7,9,13(17),14-heptaen-12-one |
|
44
|
126
|
6yqpA |
Crystal structure of the first bromodomain of human brd4 in complex with the dual inhibitor tw22 |
|
44
|
127
|
6yqoA |
Crystal structure of the first bromodomain of human brd4 in complex with the dual inhibitor tw12 |
|
45
|
125
|
6yqnA |
Crystal structure of the first bromodomain of human brd4 in complex with the dual inhibitor tw9 |
|
41
|
125
|
6xv7A |
Crystal structure of brd4-bd1 with compound 2 |
