|
40
|
113
|
5ewdA |
Crystal structure of the human brpf1 bromodomain in complex with seed18 |
|
40
|
112
|
5e3gA |
Crystal structure of the human brpf1 bromodomain in complex with seed8 |
|
41
|
112
|
5etdA |
Crystal structure of the human brpf1 bromodomain in complex with seed14 |
|
38
|
113
|
5epsA |
Crystal structure of the human brpf1 bromodomain in complex with seed10 |
|
46
|
123
|
5enjA |
Crystal structure of the second bromodomain of pleckstrin homology domain interacting protein (phip) in complex with compound-14 n11530 (sgc - diamond i04-1 fragment screening) |
|
45
|
123
|
5eneA |
Crystal structure of the second bromodomain of pleckstrin homology domain interacting protein (phip) in complex with 5-amino-2-benzyl-1,3-oxazole-4-carbonitrile (sgc - diamond i04-1 fragment screening) |
|
41
|
124
|
5eguA |
First domain of human bromodomain brd4 in complex with inhibitor 3-butyl-8-(6-butyl-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-ylsulfanylmethyl)-7-ethyl-3,7-dihydropurine-2,6-dione |
|
54
|
130
|
5f3aA |
Crystal structure of the bromodomain of human atad2 in complex with compound a14 |
|
41
|
113
|
5dycA |
Crystal structure of the human brpf1 bromodomain in complex with seed6 |
|
39
|
113
|
5dy7A |
Crystal structure of the human brpf1 bromodomain in complex with seed4 |
|
40
|
116
|
5dyuA |
Crystal structure of baz2b bromodomain in complex with fragment f39 |
|
42
|
127
|
5dlzA |
First domain of human bromodomain brd4 in complex with inhibitor 4-[(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)oxy]-n-({1-[(3-methylphe methyl]piperidin-4-yl}methyl)butanamide |
|
43
|
111
|
5dw1A |
X-ray crystal structure of human brd2(bd2) in complex with rvx297 to 1.55 a resolution |
|
38
|
116
|
5dyxA |
Crystal structure of baz2b bromodomain in complex with fragment f59 |
|
40
|
110
|
5dkcA |
Crystal structure of the bromodomain of human brm (smarca2) in complex with pfi-3 chemical probe |
|
43
|
127
|
5dw2A |
X-ray crystal structure of human brd4(bd1) in complex with rvx297 to 1.12 a resolution |
|
40
|
112
|
5dyaA |
Crystal structure of the human brpf1 bromodomain in complex with seed5 |
|
44
|
126
|
5dx4A |
Crystal structure of the first bromodomain of human brd4 in complex with benzo[cd]indol-2(1h)-one ligand |
|
41
|
109
|
5dfcA |
Crystal structure of brd2(bd2) w370f mutant with ligand i-bet 762 bound |
|
42
|
108
|
5dfdA |
Crystal structure of brd2(bd2) w370f mutant with ligand 28 bound |
|
41
|
125
|
5dlxA |
First domain of human bromodomain brd4 in complex with inhibitor n-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-1-{3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}piperidine-4-carboxamide |
|
40
|
112
|
4z93A |
Brd4 bromodomain 2 in complex with gamma-carboline-containing compound, number 18. |
|
45
|
126
|
5d24A |
First bromodomain of brd4 bound to inhibitor xd26 |
|
40
|
116
|
5dkhA |
Crystal structure of the bromodomain of human brm (smarca2) in complex with a hydroxyphenyl propenone inhibitor 17 |
|
41
|
114
|
5dbmA |
Crystal structure of the cbp bromodomain in complex with cpi703 |
|
49
|
183
|
4zqlA |
Crystal structure of trim24 with 3,4-dimethoxy-n-(6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxo-2,3-dihydro-1h-benzo[d]imidazol-5-yl)benzenesulfonamide inhibitor |
|
43
|
126
|
5d3jA |
First bromodomain of brd4 bound to inhibitor xd33 |
|
44
|
123
|
5ameA |
Crystal structure of the bromodomain of human surface epitope engineered brd1a in complex with 3d consortium fragment 4-acetyl- piperazin-2-one (sgc - diamond i04-1 fragment screening) |
|
44
|
110
|
5dkdA |
Crystal structure of the bromodomain of human brg1 (smarca4) in complex with pfi-3 chemical probe |
|
43
|
115
|
5d7xA |
Crystal structure of the human brpf1 bromodomain in complex with xz08 |
|
43
|
108
|
5dfbA |
Crystal structure of brd2(bd2) mutant w370f in the free form |
|
41
|
127
|
5d3lA |
First bromodomain of brd4 bound to inhibitor xd35 |
|
42
|
127
|
5d3tA |
First bromodomain of brd4 bound to inhibitor xd47 |
|
54
|
184
|
4yaxA |
Crystal structure of trim24 phd-bromodomain complexed with n-[6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxo-2,3-dihydro-1h-1,3-benzodiazol-5-yl]benzenesulfonamide (5g) |
|
45
|
127
|
4yh4A |
Crystal structure of human brd4(1) in complex with 4-[(5-phenylpyridin-3-yl)carbonyl]-3,4-dihydroquinoxalin-2(1h)-one (compound 19d) |
|
40
|
115
|
5cuaA |
Crystal structure of the bromodomain of bromodomain adjacent to zinc finger domain protein 2b (baz2b) in complex with 1-acetyl-4-(4-hydroxyphenyl)piperazine (sgc - diamond i04-1 fragment screening) |
|
43
|
133
|
5crmA |
Crystal structure of the first bromodomain of human brd4 in complex with benzo[cd]indol-2(1h)-one ligand |
|
44
|
126
|
5d3nA |
First bromodomain of brd4 bound to inhibitor xd40 |
|
43
|
124
|
5d25A |
First bromodomain of brd4 bound to inhibitor xd27 |
|
44
|
128
|
4yh3A |
Crystal structure of human brd4(1) in complex with 4-[(2e)-3-(4-methoxyphenyl)-2-phenylprop-2-enoyl]-3,4-dihydroquinoxalin-2(1h)-one (compound 19a) |
|
39
|
115
|
5cugA |
Crystal structure of the bromodomain of bromodomain adjacent to zinc finger domain protein 2b (baz2b) in complex with 4-acetamidobenzoic acid (sgc - diamond i04-1 fragment screening) |
|
39
|
115
|
5cq4A |
Crystal structure of the bromodomain of bromodomain adjacent to zinc finger domain protein 2b (baz2b) in complex with 3'-hydroxyacetophenone (sgc - diamond i04-1 fragment screening) |
|
42
|
115
|
5cqaA |
Crystal structure of the bromodomain of bromodomain adjacent to zinc finger domain protein 2b (baz2b) in complex with n-methyl-2,3-dihydrothieno[3,4-b][1,4]dioxine-5-carboxamide (sgc - diamond i04-1 fragment screening) |
|
43
|
125
|
5d3sA |
First bromodomain of brd4 bound to inhibitor xd44 |
|
41
|
127
|
5d3pA |
First bromodomain of brd4 bound to inhibitor xd41 |
|
50
|
183
|
4yatA |
Crystal structure of trim24 phd-bromodomain complexed with n-(1,3-dimethyl-2-oxo-2,3-dihydro-1h-1,3-benzodiazol-5-yl)-4-methoxybenzene-1-sulfonamide (5b) |
|
40
|
133
|
5ctlA |
Crystal structure of the first bromodomain of human brd4 in complex with benzo[cd]indol-2(1h)-one ligand |
|
39
|
115
|
5cudA |
Crystal structure of the bromodomain of bromodomain adjacent to zinc finger domain protein 2b (baz2b) in complex with 6-chloropurine (sgc - diamond i04-1 fragment screening) |
|
41
|
115
|
5cq7A |
Crystal structure of the bromodomain of bromodomain adjacent to zinc finger domain protein 2b (baz2b) in complex with n,n-dimethylquinoxaline-6-carboxamide (sgc - diamond i04-1 fragment screening) |
|
38
|
127
|
5d3rA |
First bromodomain of brd4 bound to inhibitor xd42 |
