|
59
|
212
|
4k4eA |
Co-crystal structure of tnks1 with compound 52 [n~2-(5-chloro-2-methoxyphenyl)-n-[trans-4-(2-oxo-2,3-dihydro-1h-benzimidazol-1-yl)cyclohexyl]glycinamide] |
|
1
|
47
|
4l32C |
Tankyrase 2 in complex with 2-[4-(4-methylpiperazine-1-carbonyl)phenyl]chromen-4-one |
|
48
|
161
|
4l0bA |
Tankyrase 2 in complex with 4'-dimethylamino flavone |
|
97
|
355
|
4l7uA |
Human artd3 (parp3) - catalytic domain in complex with inhibitor me0398 |
|
61
|
210
|
4krsA |
Tankyrase-1 complexed with small molecule inhibitor |
|
45
|
161
|
4l2gA |
Tankyrase 2 in complex with 6- fluoro flavone |
|
1
|
47
|
4l34C |
Tankyrase 2 in complex with 4'-tetrazole flavone |
|
48
|
161
|
4l33A |
Tankyrase 2 in complex with cyanomethyl 4-(4-oxo-4h-chromen-2-yl)benzoate |
|
1
|
47
|
4l0tC |
Tankyrase 2 in complex with 4'-nitro flavone |
|
113
|
357
|
4l70A |
Human artd3 (parp3) - catalytic domain in complex with inhibitor me0352 |
|
70
|
210
|
4j22A |
Tankyrase 2 in complex with 3-chloro-4-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)-n-[2-(morpholin-4-yl)ethyl]benzamide |
|
70
|
210
|
4j3mA |
Tankyrase 2 in complex with 3-chloro-4-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)benzoic acid |
|
71
|
210
|
4j21A |
Tankyrase 2 in complex with 7-(4-amino-2-chlorophenyl)-4-methylquinolin-2(1h)-one |
|
71
|
210
|
4j3lA |
Tankyrase 2 in complex with 3-chloro-n-(2-methoxyethyl)-4-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)benzamide |
|
59
|
227
|
4hyfA |
Structural basis and sar for od 270, a lead stage 1,2,4-triazole based specific tankyrase1/2 inhibitor |
|
68
|
210
|
4iueA |
Tankyrase in complex with 7-(2-fluorophenyl)-4-methyl-1,2-dihydroquinolin-2-one |
|
60
|
212
|
4i9iA |
Crystal structure of tankyrase 1 with compound 4 |
|
69
|
210
|
4j1zA |
Tankyrase 2 in complex with 4-chloro-1,2-dihydrophatalzin-one |
|
46
|
161
|
4hmhA |
Crystal structure of tankyrase 2 in complex with 7,3-dihydroxyflavone |
|
48
|
161
|
4hlfA |
Crystal structure of tankyrase 2 in complex with 7,3',4'-trihydroxyflavone |
|
48
|
161
|
4hkiA |
Tankyrase 2 in complex with flavone |
|
47
|
161
|
4hlgA |
Crystal structure of tankyrase 2 in complex with 3'-hydroxyflavone |
|
1
|
47
|
4hkiC |
Tankyrase 2 in complex with flavone |
|
1
|
47
|
4hknC |
Complex structure of human tankyrase 2 with luteolin |
|
1
|
47
|
4hlfC |
Crystal structure of tankyrase 2 in complex with 7,3',4'-trihydroxyflavone |
|
1
|
47
|
4hlhC |
Crystal structure of tankyrase 2 in complex with 4'-fluoroflavone |
|
47
|
162
|
4hkkA |
Complex structure of human tankyrase 2 with apigenin |
|
1
|
47
|
4hmhC |
Crystal structure of tankyrase 2 in complex with 7,3-dihydroxyflavone |
|
1
|
47
|
4hlkC |
Crystal structure of tankyrase 2 in complex with 4'-methylflavone |
|
1
|
47
|
4hlmC |
Crystal structure of tankyrase 2 in complex with 3',4'-dihydroxyflavone |
|
1
|
47
|
4hl5C |
Complex structure of human tankyrase 2 with 7-hydroxy -4'-methoxyflavone |
|
1
|
47
|
4hkkB |
Complex structure of human tankyrase 2 with apigenin |
|
46
|
161
|
4hlmA |
Crystal structure of tankyrase 2 in complex with 3',4'-dihydroxyflavone |
|
46
|
162
|
4hknA |
Complex structure of human tankyrase 2 with luteolin |
|
104
|
349
|
4hhzA |
Crystal structure of parp catalytic domain in complex with novel inhibitors |
|
47
|
161
|
4hlkA |
Crystal structure of tankyrase 2 in complex with 4'-methylflavone |
|
49
|
161
|
4hlhA |
Crystal structure of tankyrase 2 in complex with 4'-fluoroflavone |
|
47
|
161
|
4hl5A |
Complex structure of human tankyrase 2 with 7-hydroxy -4'-methoxyflavone |
|
106
|
349
|
4hhyA |
Crystal structure of parp catalytic domain in complex with novel inhibitors |
|
1
|
47
|
4hlgC |
Crystal structure of tankyrase 2 in complex with 3'-hydroxyflavone |
|
116
|
357
|
4gv4A |
Human artd3 (parp3) - catalytic domain in complex with inhibitor me0328 |
|
112
|
357
|
4gv2A |
Human artd3 (parp3) - catalytic domain in complex with inhibitor me0354 |
|
111
|
357
|
4gv0A |
Human artd3 (parp3) - catalytic domain in complex with inhibitor me0355 |
|
104
|
348
|
4gv7A |
Human artd1 (parp1) - catalytic domain in complex with inhibitor me0328 |
|
65
|
187
|
3q6zA |
Human parp14 (artd8)-macro domain 1 in complex with adenosine-5-diphosphoribose |
|
73
|
203
|
3q71A |
Human parp14 (artd8) - macro domain 2 in complex with adenosine-5-diphosphoribose |
|
110
|
350
|
3paxA |
The catalytic fragment of poly(adp-ribose) polymerase complexed with 3-methoxybenzamide |
|
67
|
210
|
3p0qA |
Human tankyrase 2 - catalytic parp domain in complex with an inhibitor |
|
70
|
210
|
3p0nA |
Human tankyrase 2 - catalytic parp domain in complex with an inhibitor |
|
63
|
210
|
3p0pA |
Human tankyrase 2 - catalytic parp domain in complex with an inhibitor |