|
84
|
286
|
5lvoA |
Human pdk1 kinase domain in complex with allosteric compound pse10 bound to the pif-pocket |
|
67
|
281
|
5ljjA |
Crystal structure of human mps1 (ttk) in complex with reversine |
|
83
|
274
|
5l6pA |
Ephb3 kinase domain covalently bound to an irreversible inhibitor (compound 6) |
|
88
|
284
|
5lvnA |
Human pdk1 kinase domain in complex with adenosine bound to the atp-binding site |
|
77
|
297
|
5lmkC |
Structure of phopsho-cdk2-cyclin a in complex with an atp-competitive inhibitor |
|
86
|
274
|
5l6oA |
Ephb3 kinase domain covalently bound to an irreversible inhibitor (compound 3) |
|
117
|
330
|
5m4fA |
Complex structure of human protein kinase ck2 catalytic subunit with the inhibitor 4'-carboxy-6,8-chloro-flavonol (flc21) crystallized under low-salt conditions |
|
57
|
284
|
5lohA |
Kinase domain of human greatwall |
|
112
|
347
|
5lcjA |
In-gel activity-based protein profiling of a clickable covalent erk 1/2 inhibitor |
|
88
|
276
|
5m51A |
Nek2 bound to arylaminopurine compound 8 |
|
70
|
256
|
5m09A |
Crystal structure of mycobacterium tuberculosis pkni kinase domain, c20a_r136n double mutant |
|
88
|
298
|
5l2wA |
The x-ray co-crystal structure of human cdk2/cycline and dinaciclib. |
|
78
|
276
|
5knjA |
Pseudokinase domain of mlkl bound to compound 1. |
|
68
|
292
|
5l2iA |
The x-ray co-crystal structure of human cdk6 and palbociclib. |
|
93
|
323
|
5kmnA |
Trka jm-kinase with 1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-[[2-(trifluoromethyl)phenyl]methyl]urea |
|
94
|
290
|
5l3aA |
Fragment-based discovery of 6-arylindazole jak inhibitors |
|
72
|
341
|
5kkrC |
Ksr2:mek1 complex bound to the small molecule aps-2-79 |
|
94
|
314
|
5kmmA |
Trka jm-kinase with 1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-(1-naphthyl)urea |
|
85
|
279
|
5ko1A |
Pseudokinase domain of mlkl bound to compound 4. |
|
95
|
323
|
5kmlA |
Trka jm-kinase with 1-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-3-[[2-(trifluoromethyl)phenyl]methyl]urea |
|
98
|
297
|
5kx8A |
Irak4-inhibitor co-structure |
|
90
|
315
|
5kmkA |
Trka jm-kinase with 2-fluoro-{n}-[2-(4-fluorophenyl)-6-methyl-3-pyridyl]-4-(trifluoromethyl)benzamide |
|
94
|
310
|
5kmjA |
Trka jm-kinase with {n}-(2-pyridylmethyl)-2-[2-(2-thienyl)indol-1-yl]acetamide |
|
91
|
265
|
5kupA |
Bruton's tyrosine kinase (btk) with pyridazinone compound 9 |
|
95
|
311
|
5kmiA |
Trka jm-kinase with 1-(9{h}-fluoren-9-yl)-3-(2-methyl-4-phenyl-pyrimidin-5-yl)urea |
|
80
|
291
|
5l2sA |
The x-ray co-crystal structure of human cdk6 and abemaciclib. |
|
86
|
298
|
5kmoA |
Trka jm-kinase with 1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-(2-pyridyl)urea |
|
76
|
291
|
5l2tA |
The x-ray co-crystal structure of human cdk6 and ribociclib. |
|
52
|
283
|
5kkrB |
Ksr2:mek1 complex bound to the small molecule aps-2-79 |
|
90
|
433
|
5kcvA |
Crystal structure of allosteric inhibitor, arq 092, in complex with autoinhibited form of akt1 |
|
116
|
350
|
5k4iA |
Crystal structure of erk2 in complex with compound 22 |
|
83
|
273
|
5jrqA |
Brafv600e kinase domain in complex with chemically linked vemurafenib inhibitor vem-6-vem |
|
81
|
296
|
5jq5A |
Crystal structure of cdk2 in complex with inhibitor icec0942 |
|
86
|
305
|
5jfwA |
Crystal structure of trka in complex with pf-05247452 |
|
87
|
307
|
5jgbA |
Crystal structure of human tak1/tab1 fusion protein in complex with ligand 10 |
|
90
|
287
|
5khwA |
Crystal structure of jak1 in complex with adp |
|
78
|
275
|
5k9iA |
Crystal structure of c-src in complex with a covalent lysine probe |
|
78
|
275
|
5jzjA |
Crystal structure of dclk1-kd in complex with amppn |
|
140
|
465
|
5jn2A |
Crystal structure of tgcdpk1 bound to nvpacu106 |
|
83
|
306
|
5jh6A |
Crystal structure of tl10-92 bound to tak1-tab1 |
|
85
|
305
|
5jfsA |
Crystal structure of trka in complex with pf-00593174 |
|
88
|
325
|
5j9zA |
Egfr-t790m in complex with pyrazolopyrimidine inhibitor 1a |
|
91
|
289
|
5kbqA |
Pak1 in complex with bis-anilino pyrimidine inhibitor |
|
98
|
347
|
5k5nA |
Crystal structure of gsk-3beta complexed with pf-04802367, a highly selective brain-penetrant kinase inhibitor |
|
71
|
276
|
5jt2A |
Brafv600e kinase domain in complex with chemically linked vemurafenib inhibitor vem-bisamide |
|
73
|
306
|
5jk3A |
Crystal structure of tl11-128 bound to tak1-tab1 |
|
85
|
305
|
5jfxA |
Crystal structure of trka in complex with pf-06273340 |
|
81
|
301
|
5jebA |
Crystal structure of egfr tyrosine kinase domain with novel inhibitor of active state of her2 |
|
89
|
288
|
5khxA |
Crystal structure of jak1 in complex with pf-4950736 |
|
107
|
348
|
5k5xA |
Crystal structure of human pdgfra |
