4L32C

Tankyrase 2 in complex with 2-[4-(4-methylpiperazine-1-carbonyl)phenyl]chromen-4-one
Total Genus 1
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The genus trace: a function that shows values of genus (vertical axis) for subchains spanned between the first residue, and all other residues (shown on horizontal axis). The number of the latter residue and the genus of a given subchain are shown interactively.

Total Genus
1
sequence length
47
structure length
47
Chain Sequence
MAHSPPGHHSVTGRPSVNGLALAEYVIYRGEQAYPEYLITYQIMRPE
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The genus matrix. At position (x,y) a genus value for a subchain spanned between x’th and y’th residue is shown. Values of the genus are represented by color, according to the scale given on the right.

Structure visualization

After clicking on a point (x,y) in the genus matrix above, a subchain from x to y is shown in color.

molecule tags Transferase/transferase inhibitor
molecule keywords Tankyrase-2
publication title Discovery of tankyrase inhibiting flavones with increased potency and isoenzyme selectivity.
pubmed doi rcsb
source organism Homo sapiens
total genus 1
structure length 47
sequence length 47
chains with identical sequence D
ec nomenclature ec 2.4.2.30: NAD(+) ADP-ribosyltransferase.
pdb deposition date 2013-06-05
Image from the rcsb pdb (www.rcsb.org)
cath code
ClassArchitectureTopologyHomologyDomain
3.40.1620.50 Alpha Beta 3-Layer(aba) Sandwich YefM-like fold YefM-like fold 4l32C00
4L09C 4UVPB 4HKKB 4UI8C 4L0VC 5ADSB 4L32C 4HLFC 4L2KC 4L0IC 4HKNC 4HMHC 4L0TC 4UI7C 5FPFC 4L0BC 4L0SC 4UI6C 5ADRB 4L33C 4HLMC 5ADTB 4UI3C 4KZUC 4L31C 4L34C 4HLHC 4L2FC 4UI5C 5C5PC 5C5RC 4HLKC 4L10C 4KZLC 5C5QC 4HLGC 4HL5C 4KZQC 4L2GC 4UI4C 5ADQB 4HKIC
chains in the Genus database with same CATH superfamily
4L09C 4UVPB 3CTOA 3HRYA 2ODKA 3OEIE 4HKKB 4UI8C 4L0VC 5ADSB 4L32C 3HS2A 4HLFC 4L2KC 4HKNC 4HMHC 4L0IC 4L0TC 4UI7C 5FPFC 4ZM2A 4ZM0A 3G5OA 3HJ6A 4ZLXA 4L0BC 3KH2E 4L0SC 4UI6C 5ADRB 4L33C 4HLMC 2A6QA 5ADTB 3K33B 4UI3C 4KZUC 4L31C 4L34C 3D55A 4HLHC 4L2FC 4UI5C 5C5PC 5C5RC 4HLKC 4L10C 4KZLC 5C5QC 4HLGC 3OEIA 2ZIXB 4HL5C 4KZQC 3K6QA 4L2GC 4UI4C 5ADQB 4HKIC
chains in the Genus database with same CATH topology
4L09C 4UVPB 4HKKB 4UI8C 4L0VC 5ADSB 4L32C 4HLFC 4L2KC 4L0IC 4HKNC 4HMHC 4L0TC 4UI7C 5FPFC 3HJ6A 4L0BC 4L0SC 4UI6C 5ADRB 4L33C 4HLMC 5ADTB 4UI3C 4KZUC 4L31C 4L34C 4HLHC 4L2FC 4UI5C 5C5PC 5C5RC 4HLKC 4L10C 4KZLC 5C5QC 4HLGC 4HL5C 2ZIXB 4KZQC 4L2GC 4UI4C 5ADQB 4HKIC
chains in the Genus database with same CATH homology


 
#chains in the Genus database with same CATH superfamily
 4L09 C;  4UVP B;  4HKK B;  4UI8 C;  4L0V C;  5ADS B;  4L32 C;  4HLF C;  4L2K C;  4L0I C;  4HKN C;  4HMH C;  4L0T C;  4UI7 C;  5FPF C;  4L0B C;  4L0S C;  4UI6 C;  5ADR B;  4L33 C;  4HLM C;  5ADT B;  4UI3 C;  4KZU C;  4L31 C;  4L34 C;  4HLH C;  4L2F C;  4UI5 C;  5C5P C;  5C5R C;  4HLK C;  4L10 C;  4KZL C;  5C5Q C;  4HLG C;  4HL5 C;  4KZQ C;  4L2G C;  4UI4 C;  5ADQ B;  4HKI C; 
#chains in the Genus database with same CATH topology
 4L09 C;  4UVP B;  3CTO A;  3HRY A;  2ODK A;  3OEI E;  4HKK B;  4UI8 C;  4L0V C;  5ADS B;  4L32 C;  3HS2 A;  4HLF C;  4L2K C;  4HKN C;  4HMH C;  4L0I C;  4L0T C;  4UI7 C;  5FPF C;  4ZM2 A;  4ZM0 A;  3G5O A;  3HJ6 A;  4ZLX A;  4L0B C;  3KH2 E;  4L0S C;  4UI6 C;  5ADR B;  4L33 C;  4HLM C;  2A6Q A;  5ADT B;  3K33 B;  4UI3 C;  4KZU C;  4L31 C;  4L34 C;  3D55 A;  4HLH C;  4L2F C;  4UI5 C;  5C5P C;  5C5R C;  4HLK C;  4L10 C;  4KZL C;  5C5Q C;  4HLG C;  3OEI A;  2ZIX B;  4HL5 C;  4KZQ C;  3K6Q A;  4L2G C;  4UI4 C;  5ADQ B;  4HKI C; 
#chains in the Genus database with same CATH homology
 4L09 C;  4UVP B;  4HKK B;  4UI8 C;  4L0V C;  5ADS B;  4L32 C;  4HLF C;  4L2K C;  4L0I C;  4HKN C;  4HMH C;  4L0T C;  4UI7 C;  5FPF C;  3HJ6 A;  4L0B C;  4L0S C;  4UI6 C;  5ADR B;  4L33 C;  4HLM C;  5ADT B;  4UI3 C;  4KZU C;  4L31 C;  4L34 C;  4HLH C;  4L2F C;  4UI5 C;  5C5P C;  5C5R C;  4HLK C;  4L10 C;  4KZL C;  5C5Q C;  4HLG C;  4HL5 C;  2ZIX B;  4KZQ C;  4L2G C;  4UI4 C;  5ADQ B;  4HKI C; 
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similar chains in the Genus database (?% sequence similarity)
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similar chains in the pdb database (?% sequence similarity)

 
#similar chains in the Genus database (?% sequence similarity)
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#similar chains, but unknotted
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