|
93
|
270
|
6dhaA |
Crystal structure of human ppargamma ligand binding domain in complex with hydroxy pioglitazone (m-iv) |
|
72
|
367
|
6e3sA |
Crystal structure of the heterodimeric hif-2 complex with antagonist pt2385 |
|
83
|
242
|
6owcA |
Mutant estrogen receptor alpha (era) y537s covalently bound to h3b-6545. |
|
103
|
270
|
6dgrA |
Crystal structure of human ppargamma ligand binding domain in complex with cay10638 |
|
95
|
270
|
6dh9A |
Crystal structure of human ppargamma ligand binding domain in complex with msdc-0602 |
|
100
|
270
|
6dgqA |
Crystal structure of human ppargamma ligand binding domain in complex with cay10506 |
|
97
|
270
|
6dglA |
Crystal structure of human ppargamma ligand binding domain in complex with darglitazone |
|
94
|
268
|
6dgoA |
Crystal structure of human ppargamma ligand binding domain in complex with troglitazone |
|
38
|
110
|
5jwmA |
Bivalent bet bromodomain inhibition |
|
58
|
210
|
5ke3A |
Crystal structure of setdb1 tudor domain in complex with fragment mrt0181a |
|
51
|
180
|
5h1uA |
Complex structure of trim24 phd-bromodomain and inhibitor 2 |
|
48
|
127
|
5hclA |
Crystal structure of the first bromodomain of brd4 in complex with dma |
|
50
|
182
|
5h1tA |
Complex structure of trim24 phd-bromodomain and inhibitor 1 |
|
320
|
1340
|
4yfnC |
Escherichia coli rna polymerase in complex with squaramide compound 14 (n-[3,4-dioxo-2-(4-{[4-(trifluoromethyl)benzyl]amino}piperidin-1-yl)cyclobut-1-en-1-yl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide) |
|
309
|
1369
|
4yfkD |
Escherichia coli rna polymerase in complex with squaramide compound 8. |
|
40
|
229
|
4yfxA |
Escherichia coli rna polymerase in complex with myxopyronin b |
|
23
|
89
|
4yfnE |
Escherichia coli rna polymerase in complex with squaramide compound 14 (n-[3,4-dioxo-2-(4-{[4-(trifluoromethyl)benzyl]amino}piperidin-1-yl)cyclobut-1-en-1-yl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide) |
|
39
|
112
|
6c7qA |
Brd4 bd2 in complex with compound ce277 |
|
34
|
108
|
6c7rA |
Brd4 bd1 in complex with compound cf53 |
|
82
|
228
|
6bn6A |
Identification of bicyclic hexafluoroisopropyl alcohol sulfonamides as rorgt/rorc inverse agonists |
|
85
|
240
|
5wgqA |
Estrogen receptor alpha ligand binding domain in complex with estradiol and src2-bcp1 |
|
36
|
127
|
5wmgA |
N-terminal bromodomain of brd4 in complex with otx-015 |
|
42
|
109
|
5u6vA |
X-ray crystal structure of 1,2,3-triazolobenzodiazepine in complex with brd2(d2) |
|
40
|
127
|
5wmdA |
N-terminal bromodomain of brd4 in complex with otx-015 |
|
92
|
241
|
5c4oA |
Identification of a novel allosteric binding site for rorgt inhibitors |
|
93
|
241
|
5c4tA |
Identification of a novel allosteric binding site for rorgt inhibitors |
|
317
|
1340
|
4yfkC |
Escherichia coli rna polymerase in complex with squaramide compound 8. |
|
52
|
183
|
4ybmA |
Crystal structure of trim24 phd-bromodomain complexed with n-{6-[3-(benzyloxy)phenoxy]-1,3-dimethyl-2-oxo-2,3-dihydro-1h-1,3-benzodiazol-5-yl}-3,4-dimethoxybenzene-1-sulfonamide (7b) |
|
22
|
89
|
4yfkE |
Escherichia coli rna polymerase in complex with squaramide compound 8. |
|
57
|
319
|
4yfkA |
Escherichia coli rna polymerase in complex with squaramide compound 8. |
|
57
|
183
|
4ybsA |
Crystal structure of trim24 phd-bromodomain complexed with n-{1,3-dimethyl-6-[3-(2-methylpropoxy)phenoxy]-2-oxo-2,3-dihydro-1h-1,3-benzodiazol-5-yl}-1,2-dimethyl-1h-imidazole-4-sulfonamide (7g) |
|
123
|
515
|
4yfxF |
Escherichia coli rna polymerase in complex with myxopyronin b |
|
127
|
519
|
4yfnF |
Escherichia coli rna polymerase in complex with squaramide compound 14 (n-[3,4-dioxo-2-(4-{[4-(trifluoromethyl)benzyl]amino}piperidin-1-yl)cyclobut-1-en-1-yl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide) |
|
137
|
519
|
4yfkF |
Escherichia coli rna polymerase in complex with squaramide compound 8. |
|
16
|
37
|
4u5tA |
Crystal structure of vbp leucine zipper with bound arylstibonic acid |
|
54
|
184
|
4yabA |
Crystal structure of trim24 phd-bromodomain complexed with 1-methyl-5-(2-methyl-1 3-thiazol-4-yl)-2 3-dihydro-1h-indol-2-one (1) |
|
66
|
285
|
5x54A |
Crystal structure of the keap1 kelch domain in complex with a tetrapeptide |
|
40
|
127
|
5wmaA |
N-terminal bromodomain of brd4 in complex with plx5981 |
|
1
|
11
|
5wgqE |
Estrogen receptor alpha ligand binding domain in complex with estradiol and src2-bcp1 |
|
92
|
267
|
5suxA |
Crystal structure of toxt from vibrio cholerae o395 bound to (e)-4-(8-methylnaphthalen-1-yl)but-3-enoic acid |
|
90
|
241
|
5c4uA |
Identification of a novel allosteric binding site for rorgt inhibitors |
|
92
|
241
|
5c4sA |
Identification of a novel allosteric binding site for rorgt inhibitors |
|
93
|
226
|
5k6eA |
Crystal structure of retinoic acid receptor-related orphan receptor (ror) gamma ligand binding domain complex with sbi0654919 |
|
50
|
182
|
5h1vA |
Complex structure of trim24 phd-bromodomain and inhibitor 6 |
|
43
|
127
|
5f60A |
Crystal structure of the first bromodomain of human brd4 in complex with sg3-014 |
|
40
|
127
|
5f5zA |
Crystal structure of the first bromodomain of human brd4 in complex with ma2-014 |
|
42
|
127
|
5f63A |
Crystal structure of the first bromodomain of human brd4 in complex with sg3-179 |
|
42
|
127
|
5f61A |
Crystal structure of the first bromodomain of human brd4 in complex with ma4-022-1 |
|
42
|
127
|
5f62A |
Crystal structure of the first bromodomain of human brd4 in complex with ma4-022-2 |
|
105
|
304
|
5eamA |
Crystal structure of human wdr5 in complex with compound 9o |