4BV7A

Identification of small molecule inhibitors selective for apo(a) kringles kiv-7, kiv-10 and kv.
Total Genus 22
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The genus trace: a function that shows values of genus (vertical axis) for subchains spanned between the first residue, and all other residues (shown on horizontal axis). The number of the latter residue and the genus of a given subchain are shown interactively.

Total Genus
22
sequence length
79
structure length
79
Chain Sequence
QCYHGNGQSYRGTFSTTVTGRTCQSWSSMTPHRHQRTPENYPNDGLTMNYCRNPDADTGPWCFTMDPSIRWEYCALTRC
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The genus matrix. At position (x,y) a genus value for a subchain spanned between x’th and y’th residue is shown. Values of the genus are represented by color, according to the scale given on the right.

Structure visualization

After clicking on a point (x,y) in the genus matrix above, a subchain from x to y is shown in color.

Chord Diagram
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publication title Small Molecules Used to Decipher the Pathophysiological Roles of the Kringle Domains Kiv-7, - 10 and Kv of Apolipoprotein(A)
rcsb
molecule keywords APOLIPOPROTEIN(A)
molecule tags Hydrolase
source organism Homo sapiens
total genus 22
structure length 79
sequence length 79
ec nomenclature ec 3.4.21.-:
pdb deposition date 2013-06-25

pfam database annotations

chain Pfam Accession Code Pfam Family Identifier Pfam Description
A PF00051 Kringle Kringle domain
Image from the rcsb pdb (www.rcsb.org)
cath code
ClassArchitectureTopologyHomologyDomain
2.40.20.10 Mainly Beta Beta Barrel Plasminogen Kringle 4 Plasminogen Kringle 4 4bv7A00
4BVWA 4NZQA 5CSQA 3BT2A 1KI0A 3U73A 1GMOA 5CS5A 4BVCA 4BV5A 1A0HA 1CEBA 3KIVA 1PK2A 2PF1A 4BV7A 1PMLA 1NL1A 2DOHX 5CT2A 3HN4A 3NXPA 5HPGA 1HPJA 4D3CA 2PF2A 4CIKA 5CP9A 3LAQA 1KIVA 4BVDA 5CS1A 2DOIA 4O03A 3MKPA 1NK1A 2I9AA 1GMNA 2K4RA 1I71A 1KRNA 1B2IA 2SPTA 2QJ4A 4KIVA 2K51A 2HPQP 2I9BA 1BHTA 2QJ2A 5CT3A 4BVVA 5CT1A 3E6PL 3K65A 2FEBA 2KNFA 2PK4A 2KJ4A 1PK4A 1PMKA 4HZHA 1JFNA 1PKRA 5CS9A 2FD6A 1I5KA 1HPKA 2L0SA 4A5TS 1CEAA 1NL2A 5CS3A 5COEA 4DURA 1GP9A 2HPPP 4IUAA 1TPKA 1URKA 3BT1A 3SP8A 1KDUA
chains in the Genus database with same CATH superfamily
4BVWA 4NZQA 5CSQA 3BT2A 1KI0A 3U73A 1GMOA 5CS5A 4BVCA 4BV5A 1A0HA 1CEBA 3KIVA 1PK2A 2PF1A 4BV7A 1PMLA 1NL1A 2DOHX 5CT2A 3HN4A 3NXPA 5HPGA 1HPJA 4D3CA 2PF2A 4CIKA 5CP9A 3LAQA 1KIVA 4BVDA 5CS1A 2DOIA 4O03A 3MKPA 1NK1A 2I9AA 1GMNA 2K4RA 1I71A 1KRNA 1B2IA 2SPTA 2QJ4A 4KIVA 2K51A 2HPQP 2I9BA 1BHTA 2QJ2A 5CT3A 4BVVA 5CT1A 3E6PL 3K65A 2FEBA 2KNFA 2PK4A 2KJ4A 1PK4A 1PMKA 4HZHA 1JFNA 1PKRA 5CS9A 2FD6A 1I5KA 1HPKA 2L0SA 4A5TS 1CEAA 1NL2A 5CS3A 5COEA 4DURA 1GP9A 2HPPP 4IUAA 1TPKA 1URKA 3BT1A 3SP8A 1KDUA
chains in the Genus database with same CATH topology
4BVWA 4NZQA 5CSQA 3BT2A 1KI0A 3U73A 1GMOA 5CS5A 4BVCA 4BV5A 1A0HA 1CEBA 3KIVA 1PK2A 2PF1A 4BV7A 1PMLA 1NL1A 2DOHX 5CT2A 3HN4A 3NXPA 5HPGA 1HPJA 4D3CA 2PF2A 4CIKA 5CP9A 3LAQA 1KIVA 4BVDA 5CS1A 2DOIA 4O03A 3MKPA 1NK1A 2I9AA 1GMNA 2K4RA 1I71A 1KRNA 1B2IA 2SPTA 2QJ4A 4KIVA 2K51A 2HPQP 2I9BA 1BHTA 2QJ2A 5CT3A 4BVVA 5CT1A 3E6PL 3K65A 2FEBA 2KNFA 2PK4A 2KJ4A 1PK4A 1PMKA 4HZHA 1JFNA 1PKRA 5CS9A 2FD6A 1I5KA 1HPKA 2L0SA 4A5TS 1CEAA 1NL2A 5CS3A 5COEA 4DURA 1GP9A 2HPPP 4IUAA 1TPKA 1URKA 3BT1A 3SP8A 1KDUA
chains in the Genus database with same CATH homology


 
#chains in the Genus database with same CATH superfamily
 4BVW A;  4NZQ A;  5CSQ A;  3BT2 A;  1KI0 A;  3U73 A;  1GMO A;  5CS5 A;  4BVC A;  4BV5 A;  1A0H A;  1CEB A;  3KIV A;  1PK2 A;  2PF1 A;  4BV7 A;  1PML A;  1NL1 A;  2DOH X;  5CT2 A;  3HN4 A;  3NXP A;  5HPG A;  1HPJ A;  4D3C A;  2PF2 A;  4CIK A;  5CP9 A;  3LAQ A;  1KIV A;  4BVD A;  5CS1 A;  2DOI A;  4O03 A;  3MKP A;  1NK1 A;  2I9A A;  1GMN A;  2K4R A;  1I71 A;  1KRN A;  1B2I A;  2SPT A;  2QJ4 A;  4KIV A;  2K51 A;  2HPQ P;  2I9B A;  1BHT A;  2QJ2 A;  5CT3 A;  4BVV A;  5CT1 A;  3E6P L;  3K65 A;  2FEB A;  2KNF A;  2PK4 A;  2KJ4 A;  1PK4 A;  1PMK A;  4HZH A;  1JFN A;  1PKR A;  5CS9 A;  2FD6 A;  1I5K A;  1HPK A;  2L0S A;  4A5T S;  1CEA A;  1NL2 A;  5CS3 A;  5COE A;  4DUR A;  1GP9 A;  2HPP P;  4IUA A;  1TPK A;  1URK A;  3BT1 A;  3SP8 A;  1KDU A; 
#chains in the Genus database with same CATH topology
 4BVW A;  4NZQ A;  5CSQ A;  3BT2 A;  1KI0 A;  3U73 A;  1GMO A;  5CS5 A;  4BVC A;  4BV5 A;  1A0H A;  1CEB A;  3KIV A;  1PK2 A;  2PF1 A;  4BV7 A;  1PML A;  1NL1 A;  2DOH X;  5CT2 A;  3HN4 A;  3NXP A;  5HPG A;  1HPJ A;  4D3C A;  2PF2 A;  4CIK A;  5CP9 A;  3LAQ A;  1KIV A;  4BVD A;  5CS1 A;  2DOI A;  4O03 A;  3MKP A;  1NK1 A;  2I9A A;  1GMN A;  2K4R A;  1I71 A;  1KRN A;  1B2I A;  2SPT A;  2QJ4 A;  4KIV A;  2K51 A;  2HPQ P;  2I9B A;  1BHT A;  2QJ2 A;  5CT3 A;  4BVV A;  5CT1 A;  3E6P L;  3K65 A;  2FEB A;  2KNF A;  2PK4 A;  2KJ4 A;  1PK4 A;  1PMK A;  4HZH A;  1JFN A;  1PKR A;  5CS9 A;  2FD6 A;  1I5K A;  1HPK A;  2L0S A;  4A5T S;  1CEA A;  1NL2 A;  5CS3 A;  5COE A;  4DUR A;  1GP9 A;  2HPP P;  4IUA A;  1TPK A;  1URK A;  3BT1 A;  3SP8 A;  1KDU A; 
#chains in the Genus database with same CATH homology
 4BVW A;  4NZQ A;  5CSQ A;  3BT2 A;  1KI0 A;  3U73 A;  1GMO A;  5CS5 A;  4BVC A;  4BV5 A;  1A0H A;  1CEB A;  3KIV A;  1PK2 A;  2PF1 A;  4BV7 A;  1PML A;  1NL1 A;  2DOH X;  5CT2 A;  3HN4 A;  3NXP A;  5HPG A;  1HPJ A;  4D3C A;  2PF2 A;  4CIK A;  5CP9 A;  3LAQ A;  1KIV A;  4BVD A;  5CS1 A;  2DOI A;  4O03 A;  3MKP A;  1NK1 A;  2I9A A;  1GMN A;  2K4R A;  1I71 A;  1KRN A;  1B2I A;  2SPT A;  2QJ4 A;  4KIV A;  2K51 A;  2HPQ P;  2I9B A;  1BHT A;  2QJ2 A;  5CT3 A;  4BVV A;  5CT1 A;  3E6P L;  3K65 A;  2FEB A;  2KNF A;  2PK4 A;  2KJ4 A;  1PK4 A;  1PMK A;  4HZH A;  1JFN A;  1PKR A;  5CS9 A;  2FD6 A;  1I5K A;  1HPK A;  2L0S A;  4A5T S;  1CEA A;  1NL2 A;  5CS3 A;  5COE A;  4DUR A;  1GP9 A;  2HPP P;  4IUA A;  1TPK A;  1URK A;  3BT1 A;  3SP8 A;  1KDU A; 
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